Peptide aldehyde inhibitors challenge the substrate specificity of the SARS-coronavirus main protease (Q27671833)

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11 February 2020

title

Peptide aldehyde inhibitors challenge the substrate specificity of the SARS-coronavirus main protease (English)

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11 February 2020

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inferred from abstract

structural biology

SARS-CoV-1

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based on heuristic

inferred from abstract

3C-like proteinase [SARS-Cov]

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11 February 2020

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11 February 2020

Rolf Hilgenfeld

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11 February 2020

Lili Zhu

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11 February 2020

Shyla George

series ordinal

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11 February 2020

Marco F Schmidt

series ordinal

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11 February 2020

publication date

11 August 2011

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11 February 2020

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11 February 2020

volume

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11 February 2020

issue

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11 February 2020

page(s)

204-212

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An efficient method for the synthesis of peptide aldehyde libraries employed in the discovery of reversible SARS coronavirus main protease (SARS-CoV Mpro) inhibitors

11 February 2020

cites work

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Inhibition of the severe acute respiratory syndrome 3CL protease by peptidomimetic alpha,beta-unsaturated esters

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Tripeptide aldehyde inhibitors of human rhinovirus 3C protease: design, synthesis, biological evaluation, and cocrystal structure solution of P1 glutamine isosteric replacements

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A mechanistic view of enzyme inhibition and peptide hydrolysis in the active site of the SARS-CoV 3C-like peptidase

13 September 2020

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