Facile Preparation of -Glycosylated 10-Piperazinyl Artemisinin Derivatives and Evaluation of Their Antimalarial and Cytotoxic Activities (Q56363425)

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English	Facile Preparation of -Glycosylated 10-Piperazinyl Artemisinin Derivatives and Evaluation of Their Antimalarial and Cytotoxic Activities	No description defined

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instance of

scholarly article

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title

Facile Preparation of -Glycosylated 10-Piperazinyl Artemisinin Derivatives and Evaluation of Their Antimalarial and Cytotoxic Activities (English)

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main subject

antimalarial

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glycosylation

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based on heuristic

inferred from title

author

Paola Misiano

object named as

Paola Misiano

series ordinal

4

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Donatella Taramelli

object named as

Donatella Taramelli

series ordinal

6

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Richard K Haynes

object named as

Richard K Haynes

series ordinal

8

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author name string

Yuet Wu

series ordinal

1

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Silvia Parapini

series ordinal

2

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Ian D Williams

series ordinal

3

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Ho Ning Wong

series ordinal

5

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Nicoletta Basilico

series ordinal

7

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language of work or name

English

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publication date

13 July 2018

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published in

Molecules

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volume

23

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issue

7

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copyright license

Creative Commons Attribution 4.0 International

start time

13 July 2018

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stated in

April 2022 Public Data File from Crossref

copyright status

copyrighted

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cites work

Human malaria parasites in continuous culture

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Antimalarial activity of new dihydroartemisinin derivatives. 5. Sugar analogues

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Hepatic uptake of proteins coupled to fetuin glycopeptide

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Neurotoxicity of artemisinin analogs in vitro

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stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Parasite lactate dehydrogenase as an assay for Plasmodium falciparum drug sensitivity

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Stereoelectronic properties of antimalarial artemisinin analogues in relation to neurotoxicity

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Grapefruit juice increases the bioavailability of artemether

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

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Glycosylation of fluoroquinolones through direct and oxygenated polymethylene linkages as a sugar-mediated active transport system for antimicrobials

1 reference

stated in

PubMed

reference URL

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Synthesis and biological activities of NB-506 analogues modified at the glucose group

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stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

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based on heuristic

inferred from PubMed ID database lookup

Pharmacokinetics of artemisinin-type compounds

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

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Regiocontrolled synthesis of the antitumor antibiotic AT2433-A1.

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

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inferred from PubMed ID database lookup

Efficient preparations of the beta-glucuronides of dihydroartemisinin and structural confirmation of the human glucuronide metabolite

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Neurotoxic mode of action of artemisinin

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Relative bioavailability of artesunate and dihydroartemisinin: investigations in the isolated perfused rat liver and in healthy Caucasian volunteers.

1 reference

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PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Glucuronidation of dihydroartemisinin in vivo and by human liver microsomes and expressed UDP-glucuronosyltransferases

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stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Highly Antimalaria-Active Artemisinin Derivatives: Biological Activity Does Not Correlate with Chemical Reactivity

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Galectins as modulators of tumour progression

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The pharmacokinetics of oral dihydroartemisinin and artesunate in healthy Thai volunteers.

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Structural and thermodynamic studies on cation-Pi interactions in lectin-ligand complexes: high-affinity galectin-3 inhibitors through fine-tuning of an arginine-arene interaction

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Convenient access both to highly antimalaria-active 10-arylaminoartemisinins, and to 10-alkyl ethers including artemether, arteether, and artelinate

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

4-Aminoquinoline quinolizidinyl- and quinolizidinylalkyl-derivatives with antimalarial activity

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Artemisone--a highly active antimalarial drug of the artemisinin class

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stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Molecular pharmacology and pharmacogenomics of artemisinin and its derivatives in cancer cells

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

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based on heuristic

inferred from PubMed ID database lookup

From artemisinin to new artemisinin antimalarials: biosynthesis, extraction, old and new derivatives, stereochemistry and medicinal chemistry requirements

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

In vitro activity of artemisone compared with artesunate against Plasmodium falciparum

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Galectins - potential targets for cancer therapy

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Antimalarial efficacy and drug interactions of the novel semi-synthetic endoperoxide artemisone in vitro and in vivo.

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Artesunate and dihydroartemisinin (DHA): unusual decomposition products formed under mild conditions and comments on the fitness of DHA as an antimalarial drug

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Differential effects on angiogenesis of two antimalarial compounds, dihydroartemisinin and artemisone: implications for embryotoxicity

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Anticancer properties of artemisinin derivatives and their targeted delivery by transferrin conjugation

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

First assessment in humans of the safety, tolerability, pharmacokinetics, and ex vivo pharmacodynamic antimalarial activity of the new artemisinin derivative artemisone

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

In vitro study of the anti-cancer effects of artemisone alone or in combination with other chemotherapeutic agents

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The pharmaceutical death-ride of dihydroartemisinin

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Review of the clinical pharmacokinetics of artesunate and its active metabolite dihydroartemisinin following intravenous, intramuscular, oral or rectal administration

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Antitumor activity of artemisinin and its derivatives: from a well-known antimalarial agent to a potential anticancer drug

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Anticancer properties of distinct antimalarial drug classes

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Anticancer Effect of AntiMalarial Artemisinin Compounds

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Stability of the antimalarial drug dihydroartemisinin under physiologically relevant conditions: implications for clinical treatment and pharmacokinetic and in vitro assays

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

A Randomised, Double Blind, Placebo-Controlled Pilot Study of Oral Artesunate Therapy for Colorectal Cancer

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

In vitro anti-cancer effects of artemisone nano-vesicular formulations on melanoma cells

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

In vitro skin permeation of artemisone and its nano-vesicular formulations

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Plasmodium falciparum: multifaceted resistance to artemisinins

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Fucose decorated solid-lipid nanocarriers mediate efficient delivery of methotrexate in breast cancer therapeutics.

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Methylene Homologues of Artemisone: An Unexpected Structure-Activity Relationship and a Possible Implication for the Design of C10-Substituted Artemisinins

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Emergence of Indigenous Artemisinin-Resistant Plasmodium falciparum in Africa

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identification of O-GlcNAcylated proteins in Plasmodium falciparum

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Preliminary Evaluation of Artemisinin-Cholesterol Conjugates as Potential Drugs for the Treatment of Intractable Forms of Malaria and Tuberculosis

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Synthesis, in vitro antimalarial activities and cytotoxicities of amino-artemisinin-ferrocene derivatives

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/30011856

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

DOI

10.3390/MOLECULES23071713

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PMC publication ID

6100044

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PubMed publication ID

30011856

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