Discovery and Optimization of Potent, Cell-Active Pyrazole-Based Inhibitors of Lactate Dehydrogenase (LDH). (Q47626141)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:29120638%20AND%20SRC:MED&resulttype=core&format=json

9 April 2020

title

Discovery and Optimization of Potent, Cell-Active Pyrazole-Based Inhibitors of Lactate Dehydrogenase (LDH) (English)

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9 April 2020

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9 April 2020

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9 April 2020

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9 April 2020

Leonard M Neckers

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9 April 2020

Victor M Darley-Usmar

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9 April 2020

Ganesha Rai

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9 April 2020

Kyle R Brimacombe

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9 April 2020

Bryan T Mott

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9 April 2020

Daniel J Urban

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9 April 2020

Xin Hu

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Shyh-Ming Yang

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Jennifer Kouznetsova

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Gloria A Benavides

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Katie Pohida

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9 April 2020

Eric J Kuenstner

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9 April 2020

Diane K Luci

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9 April 2020

Christine M Lukacs

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9 April 2020

Douglas R Davies

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David M Dranow

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Hu Zhu

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Gary Sulikowski

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9 April 2020

William J Moore

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9 April 2020

Gordon M Stott

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9 April 2020

Andrew J Flint

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9 April 2020

Chi V Dang

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9 April 2020

Alex G Waterson

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9 April 2020

Anton Simeonov

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9 April 2020

language of work or name

English

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publication date

9 November 2017

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Journal of Medicinal Chemistry

9 April 2020

published in

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volume

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issue

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9 April 2020

page(s)

9184-9204

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Metabolic plasticity underpins innate and acquired resistance to LDHA inhibition

9 April 2020

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Diaphorase Coupling Protocols for Red-Shifting Dehydrogenase Assays

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LDHA is necessary for the tumorigenicity of esophageal squamous cell carcinoma

29 September 2018

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29 September 2018

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29 September 2018

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29 September 2018

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29 September 2018

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29 September 2018

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1 December 2018

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1 December 2018

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12 December 2020

Hypoxia and cobalt stimulate lactate dehydrogenase (LDH) activity in vascular smooth muscle cells

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Metal binding to D-lactate dehydrogenase

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12 December 2020

10.1021/ACS.JMEDCHEM.7B00941

Identifiers

DOI

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9 April 2020

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9 April 2020

PubMed publication ID

29120638

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