Multiple conformations of 5-HT2A and 5-HT 2C receptors in rat brain: an autoradiographic study with [125I](±)DOI. (Q46899031)

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5 March 2020

title

Multiple conformations of 5-HT2A and 5-HT 2C receptors in rat brain: an autoradiographic study with [125I](±)DOI (English)

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5 March 2020

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5 March 2020

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5 March 2020

Juan F López-Giménez

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5 March 2020

José M Palacios

series ordinal

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publication date

18 July 2013

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Experimental Brain Research

5 March 2020

published in

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5 March 2020

volume

230

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issue

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5 March 2020

page(s)

395-406

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Agonist and antagonist binding to rabbit cortical 5-HT2A receptors: opposite effects of magnesium

5 March 2020

cites work

1 reference

https://api.crossref.org/works/10.1007%2FS00221-013-3636-8

A review of central 5-HT receptors and their function

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00221-013-3636-8

5-HT2 receptor subtypes: a family re-united?

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00221-013-3636-8

Evidence for distinct antagonist-revealed functional states of 5-hydroxytryptamine(2A) receptor homodimers.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00221-013-3636-8

Regulation of serotonin-2C receptor G-protein coupling by RNA editing

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00221-013-3636-8

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00221-013-3636-8

[125I]-1-(2,5-dimethoxy-4-iodophenyl)-2-amino-propane: an iodinated radioligand that specifically labels the agonist high-affinity state of 5-HT2 serotonin receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00221-013-3636-8

Functional reconstitution in situ of 5-hydroxytryptamine2c (5HT2c) receptors with alphaq and inverse agonism of 5HT2c receptor antagonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00221-013-3636-8

Serotonin receptors in the human brain. II. Characterization and autoradiographic localization of 5-HT1C and 5-HT2 recognition sites

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00221-013-3636-8

Binding to the serotonin 5-HT2 receptor by the enantiomers of 125I-DOI.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00221-013-3636-8

Agonist-receptor efficacy. II. Agonist trafficking of receptor signals

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00221-013-3636-8

SB 242084, a Selective and Brain Penetrant 5-HT 2C Receptor Antagonist

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00221-013-3636-8

Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00221-013-3636-8

Constitutive activity of receptors coupled to guanine nucleotide regulatory proteins

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00221-013-3636-8

New mouse 5-HT2-like receptor. Expression in brain, heart and intestine

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00221-013-3636-8

Common receptors for hallucinogens in rat brain: a comparative autoradiographic study using [125I]LSD and [125I]DOI, a new psychotomimetic radioligand

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00221-013-3636-8

Comparisons of hallucinogenic phenylisopropylamine binding affinities at cloned human 5-HT2A, -HT(2B) and 5-HT2C receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00221-013-3636-8

Quantitative autoradiographic mapping of serotonin receptors in the rat brain. I. Serotonin-1 receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00221-013-3636-8

Evidence for distinct 5-hydroxytryptamine2 binding site subtypes in cortical membrane preparations

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00221-013-3636-8

Distribution of the serotonin 5-HT2 receptor family mRNAs: comparison between 5-HT2A and 5-HT2C receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00221-013-3636-8

Serotonin 5-HT2A receptors: molecular biology and mechanisms of regulation

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00221-013-3636-8

G-protein coupled receptors: conformations and states

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00221-013-3636-8

Binding sites for 5-hydroxytryptamine-2 receptor agonists are predominantly located in striosomes in the human basal ganglia

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00221-013-3636-8

Antagonist functional selectivity: 5-HT2A serotonin receptor antagonists differentially regulate 5-HT2A receptor protein level in vivo

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00221-013-3636-8

Constitutively active 5-hydroxytryptamine2C receptors reveal novel inverse agonist activity of receptor ligands

21 January 2018

1 reference

12 December 2020

Pleiotropic behavior of 5-HT2A and 5-HT2C receptor agonists

1 reference

12 December 2020

Reciprocal binding properties of 5-hydroxytryptamine type 2C receptor agonists and inverse agonists

1 reference

12 December 2020

In vitro autoradiography of serotonin 5-HT2A/2C receptor-activated G protein: Guanosine-5?-(?-[35S]thio)triphosphate binding in rat brain

1 reference

12 December 2020

4-[125I]iodo-(2,5-dimethoxy)phenylisopropylamine and [3H]ketanserin labeling of 5-hydroxytryptamine2 (5HT2) receptors in mammalian cells transfected with a rat 5HT2 cDNA: evidence for multiple states and not multiple 5HT2 receptor subtypes.

1 reference

12 December 2020

International Union of Pharmacology classification of receptors for 5-hydroxytryptamine (Serotonin)

1 reference

12 December 2020

Three-state and two-state models

1 reference

12 December 2020

Molecular pharmacological differences in the interaction of serotonin with 5-hydroxytryptamine1C and 5-hydroxytryptamine2 receptors

1 reference

12 December 2020

Agonist high and low affinity state ratios predict drug intrinsic activity and a revised ternary complex mechanism at serotonin 5-HT(2A) and 5-HT(2C) receptors

1 reference

12 December 2020

Multiple conformations of native and recombinant human 5-hydroxytryptamine(2a) receptors are labeled by agonists and discriminated by antagonists.

1 reference

12 December 2020

Autoradiographic localization of binding sites for 125I-DOI, a new psychotomimetic radioligand, in the rat brain

1 reference

12 December 2020

Creation of a constitutively activated state of the 5-hydroxytryptamine2A receptor by site-directed mutagenesis: inverse agonist activity of antipsychotic drugs.

1 reference

12 December 2020

Preclinical characterization of the potential of the putative atypical antipsychotic MDL 100,907 as a potent 5-HT2A antagonist with a favorable CNS safety profile

1 reference

12 December 2020

Autoradiographic characterization of (+-)-1-(2,5-dimethoxy-4-[125I] iodophenyl)-2-aminopropane ([125I]DOI) binding to 5-HT2 and 5-HT1c receptors in rat brain.

1 reference

12 December 2020

Serotonin 5- HT (2C) receptor knockout mice: autoradiographic analysis of multiple serotonin receptors

1 reference

12 December 2020

[3H]-DOB(4-bromo-2,5-dimethoxyphenylisopropylamine) and [3H] ketanserin label two affinity states of the cloned human 5-hydroxytryptamine2 receptor

1 reference

12 December 2020

High-affinity agonist binding is not sufficient for agonist efficacy at 5-hydroxytryptamine2A receptors: evidence in favor of a modified ternary complex model

1 reference

12 December 2020

Comparative localization of serotonin1A, 1C, and2 receptor subtype mRNAs in rat brain

1 reference

12 December 2020

Multiple serotonin receptors: differential binding of [3H]5-hydroxytryptamine, [3H]lysergic acid diethylamide and [3H]spiroperidol

1 reference

12 December 2020

Differentiation of 5-hydroxytryptamine2 receptor subtypes using 125I-R-(-)2,5-dimethoxy-4-iodo-phenylisopropylamine and 3H-ketanserin.

1 reference

12 December 2020

10.1007/S00221-013-3636-8

Identifiers

DOI

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5 March 2020

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