SB 242084, a Selective and Brain Penetrant 5-HT 2C Receptor Antagonist (Q34432766)

2 August 2017

title

SB 242084, a selective and brain penetrant 5-HT2C receptor antagonist (English)

1 reference

2 August 2017

SB 242084, a Selective and Brain Penetrant 5-HT 2C Receptor Antagonist (English)

1 reference

https://api.crossref.org/works/10.1016/S0028-3908(97)00038-5

7 November 2024

G. A. Kennett

1 reference

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7 November 2024

M. D. Wood

1 reference

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7 November 2024

F. Bright

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7 November 2024

B. Trail

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7 November 2024

G. Riley

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7 November 2024

V. Holland

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7 November 2024

K. Y. Avenell

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7 November 2024

T. Stean

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7 November 2024

N. Upton

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7 November 2024

S. Bromidge

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7 November 2024

I. T. Forbes

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7 November 2024

A. M. Brown

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7 November 2024

D. N. Middlemiss

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7 November 2024

T. P. Blackburn

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7 November 2024

language of work or name

English

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National Center for Biotechnology Information

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/esummary.fcgi?db=pubmed&retmode=json&id=9225286

7 November 2024

publication date

1 April 1997

1 reference

2 August 2017

April 1997

1 reference

National Center for Biotechnology Information

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/esummary.fcgi?db=pubmed&retmode=json&id=9225286

full work available at URL

7 November 2024

number of pages

1 reference

based on heuristic

inferred from page(s)

https://api.elsevier.com/content/article/PII:S0028390897000385?httpAccept=text/xml

1 reference

https://api.crossref.org/works/10.1016/S0028-3908(97)00038-5

https://api.elsevier.com/content/article/PII:S0028390897000385?httpAccept=text/plain

7 November 2024

1 reference

https://api.crossref.org/works/10.1016/S0028-3908(97)00038-5

7 November 2024

1 reference

2 August 2017

1 reference

2 August 2017

issue

4-5

1 reference

2 August 2017

page(s)

609-620

1 reference

Cloning of another human serotonin receptor (5-HT1F): a fifth 5-HT1 receptor subtype coupled to the inhibition of adenylate cyclase

2 August 2017

cites work

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The pharmacology and distribution of human 5‐hydroxytryptamine2B (5‐HT2b) receptor gene products: comparison with 5‐HT2a and 5‐HT2c receptors

7 January 2021

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Nonlinear regression using spreadsheets.

7 January 2021

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Evidence that blockade of post-synaptic 5-HT1 receptors elicits feeding in satiated rats

7 January 2021

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Evidence for expression of the 5-hydroxytryptamine-2B receptor protein in the rat central nervous system

7 January 2021

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Activation of 5-HT 2B Receptors in the Medial Amygdala causes Anxiolysis in the Social Interaction Test in the Rat

7 January 2021

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Can social interaction be used to measure anxiety?

7 January 2021

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Increased food intake in satiated rats induced by the 5-HT antagonists methysergide, metergoline and ritanserin

7 January 2021

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The effects of chlordiazepoxide and chlorpromazine on a punishment discrimination

7 January 2021

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d-Fenfluramine- and d-norfenfluramine-induced hypophagia: differential mechanisms and involvement of postsynaptic 5-HT receptors.

7 January 2021

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Ritanserin attenuates anorectic, endocrine and thermic responses to d-fenfluramine in human volunteers.

7 January 2021

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Identification of presynaptic serotonin autoreceptors using a new ligand: 3H-PAT

7 January 2021

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Characterization of a novel 3H-5-hydroxytryptamine binding site subtype in bovine brain membranes

7 January 2021

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m-Chlorophenylpiperazine as a probe of serotonin function

7 January 2021

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Effect of SB 200646A, a 5-HT2C/5-HT2B receptor antagonist, in two conflict models of anxiety

7 January 2021

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Effects of the 5-HT2B receptor agonist, BW 723C86, on three rat models of anxiety

7 January 2021

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Evidence that hypophagia induced by mCPP and TFMPP requires 5-HT1C and 5-HT1B receptors; hypophagia induced by RU 24969 only requires 5-HT1B receptors

7 January 2021

1 reference

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In vitro and in vivo profile of SB 206553, a potent 5-HT2C/5-HT2B receptor antagonist with anxiolytic-like properties

7 January 2021

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In vivo properties of SB 200646A, a 5-HT2C/2B receptor antagonist

7 January 2021

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New mouse 5-HT2-like receptor. Expression in brain, heart and intestine

7 January 2021

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Which animal models should be used in the search for new antiepileptic drugs? A proposal based on experimental and clinical considerations

7 January 2021

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5HT2C receptor agonists exhibit antidepressant-like properties in the anhedonia model of depression in rats

7 January 2021

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(+)-cis-4,5,7a,8,9,10,11,11a-octahydro-7H-10-methylindolo[1,7- bc][2,6]-naphthyridine: a 5-HT2C/2B receptor antagonist with low 5-HT2A receptor affinity

7 January 2021

1 reference

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Distribution of the serotonin 5-HT2 receptor family mRNAs: comparison between 5-HT2A and 5-HT2C receptors

7 January 2021

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Chlorophenylpiperazine: a central serotonin agonist causing powerful anorexia in rats

7 January 2021

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Cloning and functional characterization of the human 5-HT2B serotonin receptor

7 January 2021

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Pharmacology of human dopamine D3 receptor expressed in a mammalian cell line: comparison with D2 receptor

7 January 2021

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Eating disorder and epilepsy in mice lacking 5-HT2c serotonin receptors

7 January 2021

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Characterization of alpha 1-adrenoceptor subtypes in prostate and prostatic urethra of rat, rabbit, dog and man

7 January 2021

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Characterization and distribution of putative 5-ht7 receptors in guinea-pig brain

7 January 2021

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5-HT2B receptor-mediated calcium release from ryanodine-sensitive intracellular stores in human pulmonary artery endothelial cells

7 January 2021

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Primary structure and functional characterization of a human 5-HT1D-type serotonin receptor

7 January 2021

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Molecular cloning, functional expression, and pharmacological characterization of a novel serotonin receptor (5-hydroxytryptamine2F) from rat stomach fundus

7 November 2024

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S-17-5 5HT2C receptor agonists and antagonists in animal models of anxiety

7 November 2024

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Cloning and expression of a novel serotonin receptor with high affinity for tricyclic psychotropic drugs

7 November 2024

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7 November 2024

Identifiers

1 reference

2 August 2017

1 reference