Dual targeting of DNA gyrase and topoisomerase IV: target interactions of garenoxacin (BMS-284756, T-3811ME), a new desfluoroquinolone (Q34142238)

31 July 2017

title

Dual targeting of DNA gyrase and topoisomerase IV: target interactions of garenoxacin (BMS-284756, T-3811ME), a new desfluoroquinolone (English)

1 reference

31 July 2017

Dilek Ince

1 reference

31 July 2017

Xiamei Zhang

series ordinal

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31 July 2017

L Christine Silver

series ordinal

1 reference

31 July 2017

David C Hooper

series ordinal

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31 July 2017

language of work or name

English

0 references

publication date

1 November 2002

1 reference

Antimicrobial Agents and Chemotherapy

31 July 2017

published in

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31 July 2017

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31 July 2017

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31 July 2017

page(s)

3370-3380

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NorA functions as a multidrug efflux protein in both cytoplasmic membrane vesicles and reconstituted proteoliposomes

31 July 2017

cites work

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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28 October 2018

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28 October 2018

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28 October 2018

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28 October 2018

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The mechanism of inhibition of topoisomerase IV by quinolone antibacterials

28 October 2018

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28 October 2018

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A yeast type II topoisomerase selected for resistance to quinolones. Mutation of histidine 1012 to tyrosine confers resistance to nonintercalative drugs but hypersensitivity to ellipticine.

28 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=128724

DNA gyrase-mediated wrapping of the DNA strand is required for the replication fork arrest by the DNA gyrase-quinolone-DNA ternary complex

28 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/12384338

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Mechanisms of fluoroquinolone resistance

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/12384338

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1128/AAC.46.11.3370-3380.2002

1 reference

31 July 2017

1 reference

31 July 2017

1 reference