Discovery of BI 224436, a Noncatalytic Site Integrase Inhibitor (NCINI) of HIV-1 (Q27684242)

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English	Discovery of BI 224436, a Noncatalytic Site Integrase Inhibitor (NCINI) of HIV-1	scientific article

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instance of

scholarly article

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title

Discovery of BI 224436, a Noncatalytic Site Integrase Inhibitor (NCINI) of HIV-1 (English)

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main subject

organic chemistry

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drug discovery

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HIV

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author

Anne-Marie Faucher

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31

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Eric Malenfant

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2

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Paul Edwards

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22

object named as

Paul Edwards

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author name string

Lee D Fader

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1

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Mathieu Parisien

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3

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Rebekah Carson

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4

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François Bilodeau

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5

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Serge Landry

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6

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Marc Pesant

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7

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Christian Brochu

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8

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Sébastien Morin

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9

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Catherine Chabot

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10

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Ted Halmos

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11

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Yves Bousquet

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12

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Murray D Bailey

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13

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Stephen H Kawai

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14

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René Coulombe

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15

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Steven LaPlante

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16

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Araz Jakalian

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17

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Punit K Bhardwaj

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18

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Dominik Wernic

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19

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Patricia Schroeder

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20

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Ma'an Amad

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21

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Michel Garneau

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23

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Jianmin Duan

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24

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Michael Cordingley

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25

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Richard Bethell

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26

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Stephen W Mason

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27

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Michael Bös

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28

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Pierre Bonneau

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29

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Marc-André Poupart

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30

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Bruno Simoneau

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32

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Craig Fenwick

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33

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Christiane Yoakim

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34

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Youla Tsantrizos

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35

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publication date

10 April 2014

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published in

ACS Medicinal Chemistry Letters

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stated in

Crossref

volume

5

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issue

4

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page(s)

422-7

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cites work

The A128T Resistance Mutation Reveals Aberrant Protein Multimerization as the Primary Mechanism of Action of Allosteric HIV-1 Integrase Inhibitors

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PubMed Central

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20 March 2017

Allosteric integrase inhibitor potency is determined through the inhibition of HIV-1 particle maturation

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New Class of HIV-1 Integrase (IN) Inhibitors with a Dual Mode of Action

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20 March 2017

Multimode, Cooperative Mechanism of Action of Allosteric HIV-1 Integrase Inhibitors

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20 March 2017

Rational design of small-molecule inhibitors of the LEDGF/p75-integrase interaction and HIV replication

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20 March 2017

LEDGF/p75 is essential for nuclear and chromosomal targeting of HIV-1 integrase in human cells

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20 March 2017

Identification of a small-molecule binding site at the dimer interface of the HIV integrase catalytic domain

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20 March 2017

Crystal structure of the catalytic domain of HIV-1 integrase: similarity to other polynucleotidyl transferases

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20 March 2017

Non-catalytic site HIV-1 integrase inhibitors disrupt core maturation and induce a reverse transcription block in target cells

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20 March 2017

Declining morbidity and mortality among patients with advanced human immunodeficiency virus infection. HIV Outpatient Study Investigators

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7 April 2017

Identification and characterization of a novel HIV-1 nucleotide-competing reverse transcriptase inhibitor series

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29 September 2017

The molecular biology of HIV integrase

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29 September 2017

Small-molecule inhibitors of the LEDGF/p75 binding site of integrase block HIV replication and modulate integrase multimerization

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29 September 2017

Strand transfer inhibitors of HIV-1 integrase: bringing IN a new era of antiretroviral therapy

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29 September 2017

Structural basis for the recognition between HIV-1 integrase and transcriptional coactivator p75.

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29 September 2017

Adverse effects of antiretroviral therapy

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29 September 2017

Human serum attenuates the activity of protease inhibitors toward wild-type and mutant human immunodeficiency virus

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29 September 2017

Multiple choices for HIV therapy with integrase strand transfer inhibitors

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2 June 2018

Advances in antiretroviral therapy

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27 November 2018

Grade 4 Events Are as Important as AIDS Events in the Era of HAART

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27 November 2018

HIV Drug Resistance

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reference URL

https://pubmed.ncbi.nlm.nih.gov/24900852

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

DOI

10.1021/ML500002N

1 reference

stated in

Consolidated OpenCitations Corpus – April 2017

OpenCitations bibliographic resource ID

1636970

OpenCitations bibliographic resource ID

1636970

1 reference

stated in

Consolidated OpenCitations Corpus – April 2017

OpenCitations bibliographic resource ID

1636970

PMC publication ID

4027581

1 reference

stated in

Consolidated OpenCitations Corpus – April 2017

OpenCitations bibliographic resource ID

1636970

PubMed publication ID

24900852

1 reference

stated in

Consolidated OpenCitations Corpus – April 2017

OpenCitations bibliographic resource ID

1636970

 

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