Crystal structures of the free and inhibited forms of plasmepsin I (PMI) from Plasmodium falciparum (Q27667575)

0 references

Huogen Xiao

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Takuya Miura

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Yoshiaki Kiso

Journal of Structural Biology

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language of work or name

1 reference

July 2011

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published in

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volume

175

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issue

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page(s)

73-84

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cites work

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29 September 2017

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29 September 2017

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29 September 2017

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29 September 2017

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29 September 2017

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29 September 2017

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29 September 2017

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29 September 2017

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29 September 2017

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2 June 2018

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Chipping at large, potent human T-cell leukemia virus type 1 protease inhibitors to uncover smaller, equipotent inhibitors.

27 November 2018

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27 November 2018

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X-ray structure of plasmepsin II complexed with a potent achiral inhibitor

27 November 2018

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Search for substrate-based inhibitors fitting the S2' space of malarial aspartic protease plasmepsin II.

27 November 2018

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Identification of peptidomimetic HTLV-I protease inhibitors containing hydroxymethylcarbonyl (HMC) isostere as the transition-state mimic

27 November 2018

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High-affinity inhibition of a family of Plasmodium falciparum proteases by a designed adaptive inhibitor

27 November 2018

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Biosynthesis and maturation of the malaria aspartic hemoglobinases plasmepsins I and II.

27 November 2018

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Design and synthesis of HIV protease inhibitors containing allophenylnorstatine as a transition-state mimic.

27 November 2018

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The bioavailability of oral dosage forms of a new HIV-1 protease inhibitor, KNI-272, in beagle dogs

27 November 2018

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12 December 2020

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12 December 2020

Plasmodium falciparum: differential sensitivity in vitro to E-64 (cysteine protease inhibitor) and Pepstatin A (aspartyl protease inhibitor)

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12 December 2020

Kinetic analysis of plasmepsins I and II aspartic proteases of the Plasmodium falciparum digestive vacuole

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12 December 2020

[Kynostatin (KNI)-272--a rationally designed tripeptide inhibitor of HIV protease]

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12 December 2020

Pharmacokinetic study of a tripeptide HIV-1 protease inhibitor, KNI-174, in rats after intravenous and intraduodenal administrations

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12 December 2020

10.1016/J.JSB.2011.04.009

Identifiers

DOI

1 reference

1 reference

1 reference

PubMed publication ID

21521654

1 reference