Overcoming insecticide resistance through computational inhibitor design (Q90424697)

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scientific article published on 01 October 2019

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English	Overcoming insecticide resistance through computational inhibitor design	scientific article published on 01 October 2019

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scholarly article

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Europe PubMed Central

PMC publication ID

6800356

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:31575743%20AND%20SRC:MED&resulttype=core&format=json

retrieved

13 April 2020

title

Overcoming insecticide resistance through computational inhibitor design (English)

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Europe PubMed Central

PMC publication ID

6800356

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:31575743%20AND%20SRC:MED&resulttype=core&format=json

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13 April 2020

main subject

insecticide

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based on heuristic

inferred from title

insecticide resistance

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inferred from title

author

Peter D Mabbitt

series ordinal

5

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Europe PubMed Central

PMC publication ID

6800356

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13 April 2020

Colin Jackson

series ordinal

9

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Europe PubMed Central

PMC publication ID

6800356

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:31575743%20AND%20SRC:MED&resulttype=core&format=json

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13 April 2020

Nir London

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10

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Europe PubMed Central

PMC publication ID

6800356

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:31575743%20AND%20SRC:MED&resulttype=core&format=json

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13 April 2020

Alon Harmelin

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3

object named as

Alon Harmelin

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Europe PubMed Central

PMC publication ID

6800356

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13 April 2020

Galen J Correy

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1

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Galen J Correy

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Europe PubMed Central

PMC publication ID

6800356

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:31575743%20AND%20SRC:MED&resulttype=core&format=json

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13 April 2020

author name string

Daniel Zaidman

series ordinal

2

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Europe PubMed Central

PMC publication ID

6800356

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13 April 2020

Silvia Carvalho

series ordinal

4

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PMC publication ID

6800356

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13 April 2020

Viviane Calaora

series ordinal

6

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Europe PubMed Central

PMC publication ID

6800356

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:31575743%20AND%20SRC:MED&resulttype=core&format=json

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13 April 2020

Peter J James

series ordinal

7

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Europe PubMed Central

PMC publication ID

6800356

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:31575743%20AND%20SRC:MED&resulttype=core&format=json

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13 April 2020

Andrew C Kotze

series ordinal

8

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Europe PubMed Central

PMC publication ID

6800356

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13 April 2020

publication date

1 October 2019

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Europe PubMed Central

PMC publication ID

6800356

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:31575743%20AND%20SRC:MED&resulttype=core&format=json

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13 April 2020

number of pages

10

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inferred from page(s)

published in

Proceedings of the National Academy of Sciences of the United States of America

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stated in

Europe PubMed Central

PMC publication ID

6800356

reference URL

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:31575743%20AND%20SRC:MED&resulttype=core&format=json

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13 April 2020

volume

116

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Europe PubMed Central

PMC publication ID

6800356

reference URL

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:31575743%20AND%20SRC:MED&resulttype=core&format=json

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13 April 2020

issue

42

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Europe PubMed Central

PMC publication ID

6800356

reference URL

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:31575743%20AND%20SRC:MED&resulttype=core&format=json

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13 April 2020

page(s)

21012-21021

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Europe PubMed Central

PMC publication ID

6800356

reference URL

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:31575743%20AND%20SRC:MED&resulttype=core&format=json

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13 April 2020

cites work

Gene amplification and insecticide resistance

1 reference

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PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

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inferred from PubMed ID database lookup

Mechanism of action of organophosphorus and carbamate insecticides

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stated in

PubMed

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https://pubmed.ncbi.nlm.nih.gov/31575743

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

"A" esterases and their role in regulating the toxicity of organophosphates

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PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Organophosphate poisoning

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PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

1 reference

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PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Mixed-function oxidase involvement in the biochemistry of insecticide synergists

1 reference

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PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Properties of housefly microsomal cytochromes in relation to sex, strain, substrate specificity, and apparent inhibition and induction by synergist and insecticide chemicals

1 reference

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PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

retrieved

12 December 2020

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inferred from PubMed ID database lookup

2-phenylethaneboronic acid, a possible transition-state analog for chymotrypsin

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Dieldrin and diazinon resistance in populations of the Australian sheep blowfly, Lucilia cuprina, from sheep-grazing areas and rubbish tips

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Insecticide resistance and malathion carboxylesterase in the sheep blowfly, Lucilia cuprina.

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Three distinct domains in the cholinesterase molecule confer selectivity for acetyl- and butyrylcholinesterase inhibitors

1 reference

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PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Resistance and the control of sheep ectoparasites

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

cDNA cloning, baculovirus-expression and kinetic properties of the esterase, E3, involved in organophosphorus resistance in Lucilia cuprina

1 reference

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PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

A single amino acid substitution converts a carboxylesterase to an organophosphorus hydrolase and confers insecticide resistance on a blowfly

1 reference

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PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The same amino acid substitution in orthologous esterases confers organophosphate resistance on the house fly and a blowfly

1 reference

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PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

MCE activities and malathion resistances in field populations of the australian sheep blowfly (Lucilia cuprina)

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The acetylcholinesterase gene and organophosphorus resistance in the Australian sheep blowfly, Lucilia cuprina.

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Continuous monitoring of arylesterase in human serum

1 reference

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PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Diazinon is activated by CYP2C19 in human liver

1 reference

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PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Pesticide poisoning in the developing world--a minimum pesticides list

1 reference

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PubMed

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https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Click chemistry in situ: acetylcholinesterase as a reaction vessel for the selective assembly of a femtomolar inhibitor from an array of building blocks

1 reference

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PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Boronic acid compounds as potential pharmaceutical agents

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PubMed

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https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Discovering potent and selective reversible inhibitors of enzymes in complex proteomes

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PubMed

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https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

A new and rapid colorimetric determination of acetylcholinesterase activity

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PubMed

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https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Virtual screening of chemical libraries

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PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Multiple mutations and gene duplications conferring organophosphorus insecticide resistance have been selected at the Rop-1 locus of the sheep blowfly, Lucilia cuprina

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Role of paraoxonase (PON1) status in pesticide sensitivity: genetic and temporal determinants

1 reference

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PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

A survey of mutations in the Cochliomyia hominivorax (Diptera: Calliphoridae) esterase E3 gene associated with organophosphate resistance and the molecular identification of mutant alleles.

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Multisite promiscuity in the processing of endogenous substrates by human carboxylesterase 1.

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Silencing a cotton bollworm P450 monooxygenase gene by plant-mediated RNAi impairs larval tolerance of gossypol

1 reference

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PubMed

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https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

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inferred from PubMed ID database lookup

Phasercrystallographic software

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PubMed

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https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

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XDS

1 reference

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PubMed

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https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

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PHENIX: a comprehensive Python-based system for macromolecular structure solution

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stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Features and development of Coot

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Inhibition of recombinant human carboxylesterase 1 and 2 and monoacylglycerol lipase by chlorpyrifos oxon, paraoxon and methyl paraoxon

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Functional fat body proteomics and gene targeting reveal in vivo functions of Drosophila melanogaster α-Esterase-7.

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Towards automated crystallographic structure refinement with phenix.refine

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Linking Crystallographic Model and Data Quality

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Structures of human acetylcholinesterase in complex with pharmacologically important ligands

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Inhibition of human carboxylesterases hCE1 and hiCE by cholinesterase inhibitors

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Structure and function of an insect  -carboxylesterase ( Esterase7) associated with insecticide resistance

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Better models by discarding data?

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Covalent docking of large libraries for the discovery of chemical probes

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Covalent docking predicts substrates for haloalkanoate dehalogenase superfamily phosphatases

1 reference

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PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

IRAC: Mode of action classification and insecticide resistance management

1 reference

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PubMed

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https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

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Probing questions

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PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Conformational Disorganization within the Active Site of a Recently Evolved Organophosphate Hydrolase Limits Its Catalytic Efficiency

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

retrieved

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Carboxylesterases: General detoxifying enzymes

1 reference

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PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Evolution of Protein Quaternary Structure in Response to Selective Pressure for Increased Thermostability

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Histone deacetylase enzymes as drug targets for the control of the sheep blowfly, Lucilia cuprina

1 reference

stated in

PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Mapping the Accessible Conformational Landscape of an Insect Carboxylesterase Using Conformational Ensemble Analysis and Kinetic Crystallography

1 reference

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PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

An insecticide resistance-breaking mosquitocide targeting inward rectifier potassium channels in vectors of Zika virus and malaria

1 reference

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PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Carboxylesterases in lipid metabolism: from mouse to human

1 reference

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PubMed

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https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The versatility of boron in biological target engagement

1 reference

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PubMed

reference URL

https://pubmed.ncbi.nlm.nih.gov/31575743

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12 December 2020

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Identifiers

DOI

10.1073/PNAS.1909130116

1 reference

stated in

Europe PubMed Central

PMC publication ID

6800356

reference URL

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:31575743%20AND%20SRC:MED&resulttype=core&format=json

retrieved

13 April 2020

PMC publication ID

6800356

1 reference

stated in

Europe PubMed Central

PMC publication ID

6800356

reference URL

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:31575743%20AND%20SRC:MED&resulttype=core&format=json

retrieved

13 April 2020

PubMed publication ID

31575743

1 reference

stated in

Europe PubMed Central

PMC publication ID

6800356

reference URL

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:31575743%20AND%20SRC:MED&resulttype=core&format=json

retrieved

13 April 2020

 

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