The difluoromethylenesulfonic acid group as a monoanionic phosphate surrogate for obtaining PTP1B inhibitors (Q43976130)

28 November 2017

title

The difluoromethylenesulfonic acid group as a monoanionic phosphate surrogate for obtaining PTP1B inhibitors (English)

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28 November 2017

Carmen Leung

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28 November 2017

Justyna Grzyb

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28 November 2017

Jason Lee

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28 November 2017

Natalie Meyer

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28 November 2017

Gabriel Hum

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28 November 2017

Chenguo Jia

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28 November 2017

Shifeng Liu

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28 November 2017

Scott D Taylor

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28 November 2017

language of work or name

English

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publication date

1 July 2002

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Bioorganic & Medicinal Chemistry

28 November 2017

published in

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28 November 2017

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28 November 2017

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28 November 2017

page(s)

2309-2323

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Development of inhibitors for protein tyrosine kinases

28 November 2017

cites work

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A Continuous Spectrophotometric and Fluorometric Assay for Protein Tyrosine Phosphatase Using Phosphotyrosine-Containing Peptides

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7 January 2021

Potent Inhibition of Insulin Receptor Dephosphorylation by a Hexamer Peptide Containing the Phosphotyrosyl Mimetic F2Pmp

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7 January 2021

Why is phosphonodifluoromethyl phenylalanine a more potent inhibitory moiety than phosphonomethyl phenylalanine toward protein-tyrosine phosphatases?

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7 January 2021

Affinity selection from peptide libraries to determine substrate specificity of protein tyrosine phosphatases

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Phosphonate inhibitors of protein-tyrosine and serine/threonine phosphatases

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Small molecule interactions with protein-tyrosine phosphatase PTP1B and their use in inhibitor design

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Naphthalenebis[alpha,alpha-difluoromethylenephosphonates] as potent inhibitors of protein tyrosine phosphatases

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Solid-phase synthesis of potential protein tyrosine phosphatase inhibitors via the Ugi four-component condensation

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Potent and highly selective inhibitors of the protein tyrosine phosphatase 1B

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Synthesis and biological evaluation of alpha,alpha-difluorobenzylphosphonic acid derivatives as small molecular inhibitors of protein-tyrosine phosphatase 1B

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Phosphoryltyrosyl mimetics in the design of peptide-based signal transduction inhibitors

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Examination of novel non-phosphorus-containing phosphotyrosyl mimetics against protein-tyrosine phosphatase-1B and demonstration of differential affinities toward Grb2 SH2 domains

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7 January 2021

Inhibition of protein tyrosine phosphatases PTP1B and CD45 by sulfotyrosyl peptides

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7 January 2021

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Novel phosphate mimetics for the design of non-peptidyl inhibitors of protein tyrosine phosphatases

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Synthesis of protected L-4-[sulfono(difluoromethyl)phenylalanine and its incorporation into a peptide

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Assessment of protein-tyrosine phosphatase 1B substrate specificity using "inverse alanine scanning"

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Synthesis of non-peptidyl alpha,alpha-difluoromethylenephosphonic acids on a soluble polymer support

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7 January 2021

10.1016/S0968-0896(02)00062-7

Identifiers

DOI

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28 November 2017

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