CDB-4124 and its putative monodemethylated metabolite, CDB-4453, are potent antiprogestins with reduced antiglucocorticoid activity: in vitro comparison to mifepristone and CDB-2914. (Q42519137)

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English	CDB-4124 and its putative monodemethylated metabolite, CDB-4453, are potent antiprogestins with reduced antiglucocorticoid activity: in vitro comparison to mifepristone and CDB-2914.	scientific article

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scholarly article

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Europe PubMed Central

PubMed publication ID

1 November 2017

CDB-4124 and its putative monodemethylated metabolite, CDB-4453, are potent antiprogestins with reduced antiglucocorticoid activity: in vitro comparison to mifepristone and CDB-2914. (English)

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Europe PubMed Central

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1 November 2017

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ulipristal acetate

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author name string

Barbara J Attardi

1

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Europe PubMed Central

PubMed publication ID

1 November 2017

Janet Burgenson

2

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Europe PubMed Central

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1 November 2017

Sheri A Hild

3

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Europe PubMed Central

PubMed publication ID

1 November 2017

Jerry R Reel

4

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1 November 2017

Richard P Blye

5

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1 November 2017

publication date

1 February 2002

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1 November 2017

Molecular and Cellular Endocrinology

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1 November 2017

188

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Europe PubMed Central

PubMed publication ID

1 November 2017

1-2

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Europe PubMed Central

PubMed publication ID

1 November 2017

111-123

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1 November 2017

Transcriptional regulation of the glycoprotein hormone alpha-subunit gene by pituitary adenylate cyclase-activating polypeptide (PACAP) in alphaT3-1 cells

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The progesterone antagonist RU486 acquires agonist activity upon stimulation of cAMP signaling pathways

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RU486 (mifepristone): mechanisms of action and clinical uses

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Characterization and Functional Properties of the A and B Forms of Human Progesterone Receptors Synthesized in a Baculovirus System

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CDB-2914: anti-progestational/anti-glucocorticoid profile and post-coital anti-fertility activity in rats and rabbits

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Antiovulatory and postcoital antifertility activity of the antiprogestin CDB-2914 when administered as single, multiple, or continuous doses to rats

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Identifiers

10.1016/S0303-7207(01)00743-2

1 reference

Europe PubMed Central

PubMed publication ID

1 November 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

1 November 2017

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