Interaction of positive allosteric modulators with human and Drosophila recombinant GABA receptors expressed in Xenopus laevis oocytes. (Q41991553)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8762079%20AND%20SRC:MED&resulttype=core&format=json

18 October 2019

title

Interaction of positive allosteric modulators with human and Drosophila recombinant GABA receptors expressed in Xenopus laevis oocytes (English)

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8762079%20AND%20SRC:MED&resulttype=core&format=json

18 October 2019

main subject

African clawed frog

0 references

Xenopus laevis oocyte

1 reference

1 reference

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18 October 2019

H Callachan

1 reference

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18 October 2019

C Hill-Venning

series ordinal

1 reference

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18 October 2019

J A Peters

series ordinal

1 reference

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18 October 2019

J J Lambert

series ordinal

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18 October 2019

language of work or name

English

0 references

publication date

1 June 1996

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8762079%20AND%20SRC:MED&resulttype=core&format=json

British Journal of Pharmacology

18 October 2019

published in

1 reference

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18 October 2019

volume

118

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18 October 2019

issue

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18 October 2019

page(s)

563-576

1 reference

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Pharmacological and Electrophysiological Properties of Recombinant GABAA Receptors Comprising the alpha3, beta1 and gamma2 Subunits

18 October 2019

cites work

1 reference

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Barbiturate interactions at the human GABAA receptor: dependence on receptor subunit combination

5 June 2018

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A point mutation in a Drosophila GABA receptor confers insecticide resistance.

5 June 2018

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The influence of the gamma 2L subunit on the modulation of responses to GABAA receptor activation

5 June 2018

1 reference

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Role of the beta subunit in determining the pharmacology of human gamma-aminobutyric acid type A receptors

5 June 2018

1 reference

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Propofol activates GABAA receptor-chloride ionophore complex in dissociated hippocampal pyramidal neurons of the rat.

5 June 2018

1 reference

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The modulatory action of loreclezole at the gamma-aminobutyric acid type A receptor is determined by a single amino acid in the beta 2 and beta 3 subunit

5 June 2018

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A novel allosteric modulatory site on the GABAA receptor beta subunit

5 June 2018

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Cloning and functional expression of a Drosophila gamma-aminobutyric acid receptor

5 June 2018

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Cloning and fnctional expression of an apparent splice variant of the murine 5-HT3 receptor A subunit

5 June 2018

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Pharmacology of recombinant GABAA receptors

5 June 2018

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GABAA/Benzodiazepine receptor heterogeneity: Neurophysiological implications

5 June 2018

1 reference

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Functional domains of GABAA receptors.

5 June 2018

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Potentiation, activation and blockade of GABAA receptors of clonal murine hypothalamic GT1-7 neurones by propofol.

5 June 2018

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Structure and pharmacology of gamma-aminobutyric acidA receptor subtypes.

5 June 2018

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GABAA receptor needs two homologous domains of the beta-subunit for activation by GABA but not by pentobarbital

5 June 2018

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Neurosteroids and GABAA receptor function.

5 June 2018

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Etomidate stereospecifically stimulates forebrain, but not cerebellar, 3H-diazepam binding

5 June 2018

1 reference

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Barbiturate enhancement of GABA-mediated inhibition and activation of chloride ion conductance: correlation with anticonvulsant and anesthetic actions

5 June 2018

1 reference

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Facilitatory action of etomidate and pentobarbital on recurrent inhibition in rat hippocampal pyramidal neurons

5 June 2018

1 reference

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Modulation of a GABA-ergic inhibitory circuit in the in vitro hippocampus by etomidate isomers

5 June 2018

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Modulation of the GABAA receptor by progesterone metabolites.

5 June 2018

1 reference

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Actions of pentobarbital on rat brain receptors expressed in Xenopus oocytes.

5 June 2018

1 reference

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Modulation of the GABAA receptor by depressant barbiturates and pregnane steroids

5 June 2018

1 reference

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Steroid modulation of the chloride ionophore in rat brain: structure-activity requirements, regional dependence and mechanism of action

5 June 2018

1 reference

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Steroid anesthetics and naturally occurring analogs modulate the gamma-aminobutyric acid receptor complex at a site distinct from barbiturates

5 June 2018

1 reference

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Actions of anaesthetics and avermectin on GABAA chloride channels in mammalian dorsal root ganglion neurones

5 June 2018

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Functional characteristics and sites of gene expression of the alpha 1, beta 1, gamma 2-isoform of the rat GABAA receptor

5 June 2018

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Neurochemical action of the general anaesthetic propofol on the chloride ion channel coupled with GABAA receptors

5 June 2018

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The effect of subunit composition of rat brain GABAA receptors on channel function

5 June 2018

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The actions of propofol on inhibitory amino acid receptors of bovine adrenomedullary chromaffin cells and rodent central neurones

5 June 2018

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Effects of hexachlorocyclohexanes on gamma-aminobutyric acid receptors expressed in Xenopus oocytes by RNA from mammalian brain and retina

5 June 2018

1 reference

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General anesthetics potentiate gamma-aminobutyric acid actions on gamma-aminobutyric acidA receptors expressed by Xenopus oocytes: lack of involvement of intracellular calcium

5 June 2018

1 reference

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Temperature and anion dependence of allosteric interactions at the gamma-aminobutyric acid-benzodiazepine receptor.

5 June 2018

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GABA-mimetic action of etomidate

5 June 2018

1 reference

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beta-Carboline gamma-aminobutyric acidA receptor inverse agonists modulate gamma-aminobutyric acid via the loreclezole binding site as well as the benzodiazepine site

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909744

Propofol modulates activation and desensitization of GABAA receptors in cultured murine hippocampal neurons.

18 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909744

Enhancement by propofol of the gamma-aminobutyric acidA response in dissociated hippocampal pyramidal neurons of the rat.

18 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909744

Novel properties of homomeric beta 1 gamma-aminobutyric acid type A receptors: actions of the anesthetics propofol and pentobarbital

18 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909744

Modulation of the GABAA receptor by propofol is independent of the gamma subunit.

18 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909744

Actions of the general anesthetic propofol on recombinant human GABAA receptors: influence of receptor subunits.

18 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909744

Effects of lindane (gamma-BHC) and related convulsants on GABAA receptor-operated chloride channels in frog dorsal root ganglion neurons

18 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909744

Synthesis, biological evaluation, and preliminary structure-activity considerations of a series of alkylphenols as intravenous anesthetic agents.

18 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1909744

Enhancement of Diazepam and ?-Aminobutyric Acid Binding by (+) Etomidate and Pentobarbital

18 August 2018

1 reference

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Stable expression of a functional homo-oligomeric Drosophila GABA receptor in a Drosophila cell line

18 August 2018

1 reference

Crossref

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1996.TB15439.X

Transient expression shows ligand gating and allosteric potentiation of GABAA receptor subunits

21 January 2018

1 reference

12 December 2020

Rat beta 3 subunits expressed in human embryonic kidney 293 cells form high affinity [35S]t-butylbicyclophosphorothionate binding sites modulated by several allosteric ligands of gamma-aminobutyric acid type A receptors

1 reference

12 December 2020

Single subunits of the GABAA receptor form ion channels with properties of the native receptor

1 reference

12 December 2020

Kinetic properties of the pentobarbitone-gated chloride current in frog sensory neurones

1 reference

12 December 2020

Biophysical and pharmacological properties of cloned GABAA receptor subunits expressed in Xenopus oocytes

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12 December 2020

10.1111/J.1476-5381.1996.TB15439.X

Identifiers

DOI

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8762079%20AND%20SRC:MED&resulttype=core&format=json

18 October 2019

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8762079%20AND%20SRC:MED&resulttype=core&format=json

18 October 2019

PubMed publication ID

8762079

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8762079%20AND%20SRC:MED&resulttype=core&format=json