New arylpiperazine derivatives with high affinity for alpha1A, D2 and 5-HT2A receptors (Q44249230)

1 December 2017

title

New arylpiperazine derivatives with high affinity for alpha1A, D2 and 5-HT2A receptors (English)

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1 December 2017

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1 December 2017

González-Gómez JC

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1 December 2017

Santana L

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1 December 2017

Brea J

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1 December 2017

Villazón M

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1 December 2017

Loza MI

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1 December 2017

De Luca M

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1 December 2017

Rivas ME

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1 December 2017

Montenegro GY

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1 December 2017

Fontenla JA

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1 December 2017

language of work or name

English

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publication date

1 January 2003

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Bioorganic & Medicinal Chemistry Letters

1 December 2017

published in

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1 December 2017

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1 December 2017

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1 December 2017

page(s)

175-178

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Brain Dopamine Receptors: A Primer on Their Current Status, Basic and Clinical

1 December 2017

cites work

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Short and efficient syntheses of analogues of WAY-100635: new and potent 5-HT1A receptor antagonists

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1-aryl-4-[(5-methoxy-1,2,3, 4-tetrahydronaphthalen-1-yl)alkyl]piperazines and their analogues: influence of the stereochemistry of the tetrahydronaphthalen-1-yl nucleus on 5-HT1A receptor affinity and selectivity versus alpha1 and D2 receptors. 5

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Structure-activity relationship studies of CNS agents. Part 38. Novel 1,4-benzoxazin-3(4H)-one, 1,2-benzoxazolin-3-one and 1,3-benzoxazolin-2,4-dione arylpiperazine derivatives with different 5-HT1A and antagonistic 5-HT2A activities

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7 January 2021

Effect of modifications of the alkylpiperazine moiety of trazodone on 5HT2A and alpha1 receptor binding affinity

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Synthesis and structure-activity relationships of a new model of arylpiperazines. Study of the 5-HT(1a)/alpha(1)-adrenergic receptor affinity by classical hansch analysis, artificial neural networks, and computational simulation of ligand recognitio

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Synthesis, biological evaluation, and pharmacophore generation of new pyridazinone derivatives with affinity toward alpha(1)- and alpha(2)-adrenoceptors

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Synthesis and biological activity of new 1,4-benzodioxan-arylpiperazine derivatives. Further validation of a pharmacophore model for alpha(1)-adrenoceptor antagonists

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Effects of hydralazine on contractile responses to alpha 1 and alpha 2-adrenoceptor agonists in isolated rubbed rat aorta

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New serotonin 5-HT(2A), 5-HT(2B), and 5-HT(2C) receptor antagonists: synthesis, pharmacology, 3D-QSAR, and molecular modeling of (aminoalkyl)benzo and heterocycloalkanones

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Identifiers

DOI

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release_rtv4rogoebhz7eybtb7qqyhbca

1 December 2017

Fatcat ID

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24 November 2022

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