New positron emission tomography tracer [(11)C]carvedilol reveals P-glycoprotein modulation kinetics (Q33987752)

30 July 2017

title

New positron emission tomography tracer [(11)C]carvedilol reveals P-glycoprotein modulation kinetics (English)

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positron emission tomography

30 July 2017

main subject

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Harry J M Groen

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30 July 2017

Elisabeth G.E. de Vries

object named as

Elisabeth G E de Vries

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30 July 2017

N Harry Hendrikse

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30 July 2017

Joost Bart

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30 July 2017

Eli C F Dijkers

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30 July 2017

Theodora D Wegman

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30 July 2017

Winette T A van der Graaf

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30 July 2017

Willem Vaalburg

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30 July 2017

Antoon T M Willemsen

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30 July 2017

language of work or name

English

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publication date

1 August 2005

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British Journal of Pharmacology

30 July 2017

published in

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30 July 2017

volume

145

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30 July 2017

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30 July 2017

page(s)

1045-1051

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Affinities at the verapamil binding site of MDR1-encoded P-glycoprotein: drugs and analogs, stereoisomers and metabolites

30 July 2017

cites work

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1576233

Increase in doxorubicin cytotoxicity by carvedilol inhibition of P-glycoprotein activity

28 July 2018

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A new in vivo method to study P-glycoprotein transport in tumors and the blood-brain barrier

28 July 2018

1 reference

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Complete in vivo reversal of P-glycoprotein pump function in the blood-brain barrier visualized with positron emission tomography

28 July 2018

1 reference

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Multidrug resistance: molecular mechanisms and clinical relevance

28 July 2018

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Circumvention of chemotherapy-induced myelosuppression by transfer of the mdr1 gene

28 July 2018

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Resistance-associated factors in human small-cell lung-carcinoma GLC4 sub-lines with increasing adriamycin resistance.

28 July 2018

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Relationship between lipophilicity and brain extraction of C-11-labeled radiopharmaceuticals

28 July 2018

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Graphical analysis of reversible radioligand binding from time-activity measurements applied to [N-11C-methyl]-(-)-cocaine PET studies in human subjects

28 July 2018

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Quantitative assessment of P-glycoprotein function in the rat blood-brain barrier by distribution volume of [11C]verapamil measured with PET.

28 July 2018

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Increased 99mTc-sestamibi accumulation in normal liver and drug-resistant tumors after the administration of the glycoprotein inhibitor, XR9576.

29 October 2018

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Synthesis and evaluation of radiolabeled antagonists for imaging of beta-adrenoceptors in the brain with PET.

29 October 2018

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Benefit of cyclosporine modulation of drug resistance in patients with poor-risk acute myeloid leukemia: a Southwest Oncology Group study

29 October 2018

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Phase I and pharmacokinetic study of the novel MDR1 and MRP1 inhibitor biricodar administered alone and in combination with doxorubicin

29 October 2018

1 reference

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Graphical analysis of PET data applied to reversible and irreversible tracers

29 October 2018

1 reference

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Quantitative ex vivo and in vitro receptor autoradiography using 11C-labeled ligands and an imaging plate: a study with a dopamine D2-like receptor ligand [11C]nemonapride

29 October 2018

1 reference

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Treatment of refractory and relapsed acute myelogenous leukemia with combination chemotherapy plus the multidrug resistance modulator PSC 833 (Valspodar).

29 October 2018

1 reference

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Octanol-water partition: searching for predictive models

29 October 2018

1 reference

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Metabolism of carvedilol in man

29 October 2018

1 reference

12 December 2020

Receptor imaging technique with 11C-labeled receptor ligands in living brain slices: its application to time-resolved imaging and saturation analysis of benzodiazepine receptor using [11C]Ro15-1788

1 reference

12 December 2020

Modulation of the multidrug resistance P-glycoprotein: detection with technetium-99m-sestamibi in vivo

1 reference

12 December 2020

Methodological aspects for in vitro characterization of receptor binding using 11C-labeled receptor ligands: A detailed study with the benzodiazepine receptor antagonist [11C]Ro 15-1788

1 reference

12 December 2020

Metabolism of carvedilol in dogs, rats, and mice

1 reference

12 December 2020

Detection of in vivo P-glycoprotein inhibition by PSC 833 using Tc-99m sestamibi

1 reference

12 December 2020

Identifiers

DOI

10.1038/SJ.BJP.0706283

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30 July 2017

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30 July 2017

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