Novel positive allosteric modulators of GABAA receptors: do subtle differences in activity at alpha1 plus alpha5 versus alpha2 plus alpha3 subunits account for dissimilarities in behavioral effects in rats? (Q33810376)

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English	Novel positive allosteric modulators of GABAA receptors: do subtle differences in activity at alpha1 plus alpha5 versus alpha2 plus alpha3 subunits account for dissimilarities in behavioral effects in rats?	scientific article

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scholarly article

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29 July 2017

Novel positive allosteric modulators of GABAA receptors: do subtle differences in activity at alpha1 plus alpha5 versus alpha2 plus alpha3 subunits account for dissimilarities in behavioral effects in rats? (English)

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29 July 2017

author name string

Miroslav M Savić

1

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29 July 2017

Samarpan Majumder

2

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29 July 2017

Shengming Huang

3

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29 July 2017

Rahul V Edwankar

4

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29 July 2017

Roman Furtmüller

5

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29 July 2017

Srdan Joksimović

6

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29 July 2017

Terry Clayton

7

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29 July 2017

Joachim Ramerstorfer

8

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29 July 2017

Marija M Milinković

9

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29 July 2017

Bryan L Roth

10

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29 July 2017

Werner Sieghart

11

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29 July 2017

James M Cook

12

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29 July 2017

publication date

13 January 2010

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29 July 2017

Progress in Neuro-Psychopharmacology & Biological Psychiatry

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29 July 2017

34

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29 July 2017

2

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29 July 2017

376-386

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29 July 2017

Target site occupancy: emerging generalizations from clinical and preclinical studies

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Antiseizure activity of novel gamma-aminobutyric acid (A) receptor subtype-selective benzodiazepine analogues in mice and rat models

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GABA-A receptors: a viable target for novel anxiolytics?

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Selective anxiolysis produced by ocinaplon, a GABA(A) receptor modulator.

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Positioning of the alpha-subunit isoforms confers a functional signature to gamma-aminobutyric acid type A receptors.

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Cloning of cDNA sequences encoding human alpha 2 and alpha 3 gamma-aminobutyric acidA receptor subunits and characterization of the benzodiazepine pharmacology of recombinant alpha 1-, alpha 2-, alpha 3-, and alpha 5-containing human [...]

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Diazepam impairs acquisition but not performance in the Morris water maze

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The effect of subunit composition of rat brain GABAA receptors on channel function

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A single histidine in GABAA receptors is essential for benzodiazepine agonist binding

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Research in anxiety disorders: from the bench to the bedside

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Molecular basis for the GABAA receptor-mediated tonic inhibition in rat somatosensory cortex

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12 December 2020

based on heuristic

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Benzodiazepine site inverse agonists and locomotor activity in rats: bimodal and biphasic influence

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12 December 2020

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10.1016/J.PNPBP.2010.01.004

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Europe PubMed Central

PubMed publication ID

29 July 2017

PMC publication ID

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Europe PubMed Central

PubMed publication ID

29 July 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

29 July 2017

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