Comprehensive characterization of cytochrome P450 isozyme selectivity across chemical libraries (Q33512310)

27 July 2017

title

Comprehensive characterization of cytochrome P450 isozyme selectivity across chemical libraries (English)

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27 July 2017

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27 July 2017

Darren Fayne

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David G Lloyd

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Christopher P Austin

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27 July 2017

Douglas S Auld

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27 July 2017

Henrike Veith

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27 July 2017

Ruili Huang

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27 July 2017

Tim James

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27 July 2017

Natalia Artemenko

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27 July 2017

Min Shen

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27 July 2017

James Inglese

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27 July 2017

publication date

25 October 2009

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27 July 2017

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27 July 2017

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27 July 2017

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27 July 2017

page(s)

1050-1055

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Identification of pregnane X receptor ligands using time-resolved fluorescence resonance energy transfer and quantitative high-throughput screening

27 July 2017

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31 October 2018

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31 October 2018

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31 October 2018

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31 October 2018

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31 October 2018

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12 December 2020

Structural determinants of cytochrome P450 substrate specificity, binding affinity and catalytic rate

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12 December 2020

CYP2C9 inhibition: impact of probe selection and pharmacogenetics on in vitro inhibition profiles

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12 December 2020

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12 December 2020

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12 December 2020

Identifiers

DOI

10.1038/NBT.1581

1 reference

27 July 2017

1 reference

27 July 2017

1 reference