A high-throughput cell-based assay for inhibitors of ABCG2 activity (Q33234390)

24 July 2017

title

A high-throughput cell-based assay for inhibitors of ABCG2 activity (English)

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24 July 2017

Michael Dean

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Robert W Robey

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Susan E Bates

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24 July 2017

Curtis J Henrich

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24 July 2017

Heidi R Bokesch

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24 July 2017

Ekaterina I Goncharova

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24 July 2017

Jennifer A Wilson

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24 July 2017

James B McMahon

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24 July 2017

publication date

20 February 2006

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Journal of Biomolecular Screening

24 July 2017

published in

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24 July 2017

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24 July 2017

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24 July 2017

page(s)

176-183

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Mammalian ABC transporters in health and disease

24 July 2017

cites work

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https://api.crossref.org/works/10.1177%2F1087057105284576

The human ATP-binding cassette (ABC) transporter superfamily

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105284576

Multidrug resistance mediated by the breast cancer resistance protein BCRP (ABCG2)

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105284576

Tumour stem cells and drug resistance

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105284576

Interaction of the breast cancer resistance protein with plant polyphenols

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105284576

The breast cancer resistance protein protects against a major chlorophyll-derived dietary phototoxin and protoporphyria.

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105284576

Frequent expression of the multi-drug resistance-associated protein BCRP/MXR/ABCP/ABCG2 in human tumours detected by the BXP-21 monoclonal antibody in paraffin-embedded material

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105284576

Increased oral bioavailability of topotecan in combination with the breast cancer resistance protein and P-glycoprotein inhibitor GF120918.

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105284576

ABCG2 (BCRP) expression in normal and malignant hematopoietic cells

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105284576

Pheophorbide a is a specific probe for ABCG2 function and inhibition.

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105284576

Mammalian drug efflux transporters of the ATP binding cassette (ABC) family: an overview.

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105284576

A functional assay for detection of the mitoxantrone resistance protein, MXR (ABCG2).

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105284576

Effects of dihydropyridines and pyridines on multidrug resistance mediated by breast cancer resistance protein: in vitro and in vivo studies

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105284576

A Simple Statistical Parameter for Use in Evaluation and Validation of High Throughput Screening Assays

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105284576

Functional characterization of the human multidrug transporter, ABCG2, expressed in insect cells

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105284576

Characterization of drug transport, ATP hydrolysis, and nucleotide trapping by the human ABCG2 multidrug transporter. Modulation of substrate specificity by a point mutation

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105284576

Differential sensitivities of the human ATP-binding cassette transporters ABCG2 and P-glycoprotein to cyclosporin A.

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105284576

Reversal of breast cancer resistance protein (BCRP/ABCG2)‐mediated drug resistance by novobiocin, a coumermycin antibiotic

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105284576

Mutations at amino-acid 482 in the ABCG2 gene affect substrate and antagonist specificity.

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105284576

Flavonoids are inhibitors of breast cancer resistance protein (ABCG2)-mediated transport

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105284576

The ABC transporter Bcrp1/ABCG2 is expressed in a wide variety of stem cells and is a molecular determinant of the side-population phenotype

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105284576

Synergistic antitumor effect of combined use of adenoviral-mediated p53 gene transfer and antisense oligodeoxynucleotide targeting clusterin gene in an androgen-independent human prostate cancer model.

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105284576

Flow cytometry-based approach to ABCG2 function suggests that the transporter differentially handles the influx and efflux of drugs

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105284576

Flavonoid structure-activity studies identify 6-prenylchrysin and tectochrysin as potent and specific inhibitors of breast cancer resistance protein ABCG2.

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105284576

Structure activity relationships and quantitative structure activity relationships for the flavonoid-mediated inhibition of breast cancer resistance protein

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105284576

VX-710 (biricodar) increases drug retention and enhances chemosensitivity in resistant cells overexpressing P-glycoprotein, multidrug resistance protein, and breast cancer resistance protein

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105284576

Broad-spectrum modulation of ATP-binding cassette transport proteins by the taxane derivatives ortataxel (IDN-5109, BAY 59-8862) and tRA96023.

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105284576

21 January 2018

Identifiers

DOI

10.1177/1087057105284576

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24 July 2017

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