Design, synthesis, and discovery of 3-piperazinyl-3,4-dihydro-2(1H)-quinolinone derivatives: a novel series of mixed dopamine D2/D4 receptor antagonists (Q31440471)

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English	Design, synthesis, and discovery of 3-piperazinyl-3,4-dihydro-2(1H)-quinolinone derivatives: a novel series of mixed dopamine D2/D4 receptor antagonists	scientific article

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scholarly article

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Europe PubMed Central

PubMed publication ID

2 July 2017

Design, synthesis, and discovery of 3-piperazinyl-3,4-dihydro-2(1H)-quinolinone derivatives: a novel series of mixed dopamine D2/D4 receptor antagonists (English)

1 reference

Europe PubMed Central

PubMed publication ID

2 July 2017

author name string

Zhao H

1

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Europe PubMed Central

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2 July 2017

Thurkauf A

2

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Europe PubMed Central

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2 July 2017

Braun J

3

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Europe PubMed Central

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2 July 2017

Brodbeck R

4

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2 July 2017

Kieltyka A

5

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2 July 2017

language of work or name

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publication date

1 September 2000

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2 July 2017

Bioorganic & Medicinal Chemistry Letters

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2 July 2017

10

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PubMed publication ID

2 July 2017

18

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Europe PubMed Central

PubMed publication ID

2 July 2017

2119-2122

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Europe PubMed Central

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2 July 2017

Dopamine receptor pharmacology

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Molecular cloning and expression of the gene for a human D1 dopamine receptor

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Cloning of the gene for a human dopamine D5 receptor with higher affinity for dopamine than D1

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Cloning and expression of a rat D2 dopamine receptor cDNA

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Cloning of the gene for a human dopamine D4 receptor with high affinity for the antipsychotic clozapine

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D4 receptors and their antagonists

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Isoindolinone enantiomers having affinity for the dopamine D4 receptor

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(S)-(-)-4-[4-[2-(isochroman-1-yl)ethyl]-piperazin-1-yl] benzenesulfonamide, a selective dopamine D4 antagonist

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Synthesis, SAR and pharmacology of CP-293,019: a potent, selective dopamine D4 receptor antagonist

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Centrally acting dopamine D2 receptor ligands: agonists

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New generation dopaminergic agents. 6. Structure-activity relationship studies of a series of 4-(aminoethoxy)indole and 4-(aminoethoxy)indolone derivatives based on the newly discovered 3-hydroxyphenoxyethylamine D2 template

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Identifiers

10.1016/S0960-894X(00)00421-2

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Europe PubMed Central

PubMed publication ID

2 July 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

2 July 2017

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