Impact of D2 receptor internalization on binding affinity of neuroimaging radiotracers. (Q39768071)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:19956086%20AND%20SRC:MED&resulttype=core&format=json

13 February 2020

title

Impact of D2 receptor internalization on binding affinity of neuroimaging radiotracers (English)

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13 February 2020

0 references

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13 February 2020

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13 February 2020

Ningning Guo

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13 February 2020

Wen Guo

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13 February 2020

Michaela Kralikova

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13 February 2020

Man Jiang

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13 February 2020

Ira Schieren

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13 February 2020

Raj Narendran

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13 February 2020

Mark Slifstein

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13 February 2020

Marc Laruelle

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13 February 2020

Anissa Abi-Dargham

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13 February 2020

language of work or name

English

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publication date

2 December 2009

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13 February 2020

published in

Neuropsychopharmacology

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13 February 2020

volume

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13 February 2020

issue

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13 February 2020

page(s)

806-817

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G protein-coupled receptor kinase-mediated phosphorylation regulates post-endocytic trafficking of the D2 dopamine receptor.

13 February 2020

cites work

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Small effect of dopamine release and no effect of dopamine depletion on [18F]fallypride binding in healthy humans

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A cysteine residue in the third membrane-spanning segment of the human D2 dopamine receptor is exposed in the binding-site crevice.

22 September 2017

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Comparison of three high affinity SPECT radiotracers for the dopamine D2 receptor

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15 June 2018

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Preparation of [76Br]FLB 457 and [76Br]FLB 463 for examination of striatal and extrastriatal dopamine D-2 receptors with PET.

15 June 2018

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20 August 2018

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20 August 2018

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20 August 2018

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20 August 2018

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20 August 2018

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20 August 2018

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20 August 2018

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Radiosynthesis and evaluation of [11C]-(+)-4-propyl-3,4,4a,5,6,10b-hexahydro-2H-naphtho[1,2-b][1,4]oxazin-9-ol as a potential radiotracer for in vivo imaging of the dopamine D2 high-affinity state with positron emission tomography.

20 August 2018

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20 August 2018

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20 August 2018

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20 August 2018

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20 August 2018

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Effect of endogenous dopamine on extrastriatal [¹¹C]FLB 457 binding measured by PET.

20 August 2018

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20 August 2018

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Imaging D2 receptor occupancy by endogenous dopamine in humans

20 August 2018

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20 August 2018

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Regional distribution of sultopride and sulpiride in rat brain measured by radioimmunoassay

20 August 2018

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Striatal D1- and D2-dopamine receptor sites are separately detectable in vivo

20 August 2018

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Endogenous dopamine (DA) modulates [3H]spiperone binding in vivo in rat brain

20 August 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/19956086

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Amphetamine effects on dopamine release and synthesis rate studied in the Rhesus monkey brain by positron emission tomography

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/19956086

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Sequestration of dopamine D2 receptors depends on coexpression of G-protein-coupled receptor kinases 2 or 5

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/19956086

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1038/NPP.2009.189

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:19956086%20AND%20SRC:MED&resulttype=core&format=json

13 February 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:19956086%20AND%20SRC:MED&resulttype=core&format=json

13 February 2020

PubMed publication ID

19956086

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:19956086%20AND%20SRC:MED&resulttype=core&format=json