Macrocyclic peptoid-Peptide hybrids as inhibitors of class I histone deacetylases. (Q39735346)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24900543%20AND%20SRC:MED&resulttype=core&format=json

20 March 2020

title

Macrocyclic peptoid-Peptide hybrids as inhibitors of class I histone deacetylases (English)

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20 March 2020

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20 March 2020

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20 March 2020

Ana Montero

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20 March 2020

M Reza Ghadiri

series ordinal

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20 March 2020

publication date

10 August 2012

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ACS Medicinal Chemistry Letters

20 March 2020

published in

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20 March 2020

volume

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20 March 2020

issue

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20 March 2020

page(s)

749-753

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Discovery of HDAC Inhibitors That Lack an Active Site Zn(2+)-Binding Functional Group.

20 March 2020

cites work

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Potential Agents for Treating Cystic Fibrosis: Cyclic Tetrapeptides that Restore Trafficking and Activity of ΔF508-CFTR

14 September 2017

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Extraordinarily robust polyproline type I peptoid helices generated via the incorporation of α-chiral aromatic N-1-naphthylethyl side chains

14 September 2017

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14 September 2017

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Inside HDAC with HDAC inhibitors

14 September 2017

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14 September 2017

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14 September 2017

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Discovery of potent and selective histone deacetylase inhibitors via focused combinatorial libraries of cyclic alpha3beta-tetrapeptides

14 September 2017

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Peptoids as potential therapeutics.

14 September 2017

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Probing the bioactive conformation of an archetypal natural product HDAC inhibitor with conformationally homogeneous triazole-modified cyclic tetrapeptides.

14 September 2017

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Conformationally homogeneous heterocyclic pseudotetrapeptides as three-dimensional scaffolds for rational drug design: receptor-selective somatostatin analogues

14 September 2017

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Design, synthesis, biological evaluation, and structural characterization of potent histone deacetylase inhibitors based on cyclic alpha/beta-tetrapeptide architectures.

14 September 2017

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Design and synthesis of macrocyclic peptomers as mimics of a quorum sensing signal from Staphylococcus aureus

14 September 2017

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A peptoid "antibody surrogate" that antagonizes VEGF receptor 2 activity

14 September 2017

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From natural products to small molecule ketone histone deacetylase inhibitors: development of new class specific agents

14 September 2017

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Peptoids that mimic the structure, function, and mechanism of helical antimicrobial peptides

14 September 2017

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Histone deacetylase inhibitors: from bench to clinic

14 September 2017

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Dimethyl sulfoxide to vorinostat: development of this histone deacetylase inhibitor as an anticancer drug

14 September 2017

1 reference

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Anticancer activities of histone deacetylase inhibitors

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025818

Histone deacetylase inhibitors and the promise of epigenetic (and more) treatments for cancer

14 September 2017

1 reference

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Epigenetics--an epicenter of gene regulation: histones and histone-modifying enzymes

14 September 2017

1 reference

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Exploiting the basis of proline recognition by SH3 and WW domains: design of N-substituted inhibitors

14 September 2017

1 reference

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Apicidin: a novel antiprotozoal agent that inhibits parasite histone deacetylase

14 September 2017

1 reference

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Peptoids: a modular approach to drug discovery.

14 September 2017

1 reference

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The activity of HDAC8 depends on local and distal sequences of its peptide substrates

14 September 2017

1 reference

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A conformationally frozen peptoid boosts CXCR4 affinity and anti-HIV activity

17 June 2018

1 reference

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Design, synthesis and antimicrobial properties of non-hemolytic cationic alpha-cyclopeptoids

20 August 2018

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Antimicrobial beta-peptoids by a block synthesis approach.

20 August 2018

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Solution, solid phase and computational structures of apicidin and its backbone-reduced analogs

20 August 2018

1 reference

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Molecular evolution of the histone deacetylase family: functional implications of phylogenetic analysis.

20 August 2018

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FK228 (depsipeptide) as a natural prodrug that inhibits class I histone deacetylases

20 August 2018

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The Click Triazolium Peptoid Side Chain: A Strong cis-Amide Inducer Enabling Chemical Diversity

20 August 2018

1 reference

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Antiplasmodial and Prehemolytic Activities of α-Peptide–β-Peptoid Chimeras

1 October 2018

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12 December 2020

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12 December 2020

Alpha-peptide/beta-peptoid chimeras

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12 December 2020

Antimicrobial, Hemolytic, and Cytotoxic Activities of β-Peptoid-Peptide Hybrid Oligomers: Improved Properties Compared to Natural AMPs

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12 December 2020

Probing the structural requirements of peptoids that inhibit HDM2-p53 interactions

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12 December 2020

A comparison of linear and cyclic peptoid oligomers as potent antimicrobial agents

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12 December 2020

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12 December 2020

Identifiers

DOI

10.1021/ML300162R

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24900543%20AND%20SRC:MED&resulttype=core&format=json

20 March 2020

1 reference

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20 March 2020

PubMed publication ID

24900543

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24900543%20AND%20SRC:MED&resulttype=core&format=json