Allosteric modulation, thermodynamics and binding to wild-type and mutant (T277A) adenosine A1 receptors of LUF5831, a novel nonadenosine-like agonist (Q38756711)

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scientific article published on March 2006

Language	Label	Description	Also known as
English	Allosteric modulation, thermodynamics and binding to wild-type and mutant (T277A) adenosine A1 receptors of LUF5831, a novel nonadenosine-like agonist	scientific article published on March 2006

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scholarly article

1 reference

Europe PubMed Central

PMC publication ID

6 September 2017

Allosteric modulation, thermodynamics and binding to wild-type and mutant (T277A) adenosine A1 receptors of LUF5831, a novel nonadenosine-like agonist (English)

1 reference

Europe PubMed Central

PMC publication ID

6 September 2017

Laura H Heitman

object named as

Laura H Heitman

1

0 references

Adriaan P IJzerman

object named as

Adriaan P IJzerman

6

0 references

author name string

Thea Mulder-Krieger

2

1 reference

Europe PubMed Central

PMC publication ID

6 September 2017

Ronald F Spanjersberg

3

1 reference

Europe PubMed Central

PMC publication ID

6 September 2017

Jacobien K von Frijtag Drabbe Künzel

4

1 reference

Europe PubMed Central

PMC publication ID

6 September 2017

Alessandro Dalpiaz

5

1 reference

Europe PubMed Central

PMC publication ID

6 September 2017

language of work or name

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publication date

1 March 2006

1 reference

Europe PubMed Central

PMC publication ID

6 September 2017

British Journal of Pharmacology

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Europe PubMed Central

PMC publication ID

6 September 2017

147

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Europe PubMed Central

PMC publication ID

6 September 2017

5

1 reference

Europe PubMed Central

PMC publication ID

6 September 2017

533-541

1 reference

Europe PubMed Central

PMC publication ID

6 September 2017

Effects of the allosteric modulator SCH-202676 on adenosine and P2Y receptors

1 reference

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6 September 2017

Receptor binding thermodynamics at the neuronal nicotinic receptor

1 reference

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Medicinal chemistry of adenosine A1 receptor ligands

1 reference

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International Union of Pharmacology. XXV. Nomenclature and classification of adenosine receptors

1 reference

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A1 adenosine receptors and their ligands: overview and recent developments

1 reference

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Differential effects of the allosteric enhancer (2-amino-4,5-dimethyl-trienyl)[3-trifluoromethyl) phenyl]methanone (PD81,723) on agonist and antagonist binding and function at the human wild-type and a mutant (T277A) adenosine A1 receptor

1 reference

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1 reference

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Thermodynamics of full agonist, partial agonist, and antagonist binding to wild-type and mutant adenosine A1 receptors.

1 reference

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A threonine residue in the seventh transmembrane domain of the human A1 adenosine receptor mediates specific agonist binding

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Synthesis and biological evaluation of a new series of 2,3,5-substituted [1,2,4]-thiadiazoles as modulators of adenosine A1 receptors and their molecular mechanism of action

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1 reference

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1 reference

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1 reference

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Partial agonism of theophylline-7-riboside on adenosine receptors

1 reference

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PD 81,723, an allosteric enhancer of the A1 adenosine receptor, lowers the threshold for ischemic preconditioning in dogs

1 reference

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Agonist-independent effect of an allosteric enhancer of the A1 adenosine receptor in CHO cells stably expressing the recombinant human A1 receptor

1 reference

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12 December 2020

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Identifiers

10.1038/SJ.BJP.0706655

1 reference

Europe PubMed Central

PMC publication ID

6 September 2017

PMC publication ID

1 reference

Europe PubMed Central

PMC publication ID

6 September 2017

PubMed publication ID

1 reference

Europe PubMed Central

PMC publication ID

6 September 2017

ResearchGate publication ID

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