In vitro and in vivo pharmacological profile of UFP-512, a novel selective delta-opioid receptor agonist; correlations between desensitization and tolerance. (Q36358677)

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English	In vitro and in vivo pharmacological profile of UFP-512, a novel selective delta-opioid receptor agonist; correlations between desensitization and tolerance.	scientific article

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scholarly article

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9 January 2020

In vitro and in vivo pharmacological profile of UFP-512, a novel selective delta-opioid receptor agonist; correlations between desensitization and tolerance (English)

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9 January 2020

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desensitization

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based on heuristic

inferred from title

Severo Salvadori

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9 January 2020

Stéphane Allouche

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9 January 2020

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B Aguila

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L Coulbault

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9 January 2020

M Boulouard

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F Léveillé

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9 January 2020

A Davis

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G Tóth

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A Borsodi

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G Balboni

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P Jauzac

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5 November 2007

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9 January 2020

British Journal of Pharmacology

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9 January 2020

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9 January 2020

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9 January 2020

1312-1324

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9 January 2020

High-purity selection and maintenance of gene expression in human neuroblastoma cells stably over-expressing GFP fusion protein. Application for opioid receptors desensitization studies

1 reference

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30 September 2017

Distinct signaling profiles of beta1 and beta2 adrenergic receptor ligands toward adenylyl cyclase and mitogen-activated protein kinase reveals the pluridimensionality of efficacy

1 reference

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30 September 2017

The antidepressant -like effects of delta-opioid receptor agonists

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30 September 2017

Tracking the opioid receptors on the way of desensitization

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30 September 2017

Morphine promotes rapid, arrestin-dependent endocytosis of mu-opioid receptors in striatal neurons

1 reference

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30 September 2017

Different regulation of human delta-opioid receptors by SNC-80 [(+)-4-[(alphaR)-alpha-((2S,5R)-4-allyl-2,5-dimethyl-1-piperazinyl)-3-methoxybenzyl]-N,N-diethylbenzamide] and endogenous enkephalins.

1 reference

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30 September 2017

Pharmacological characterization of AR-M1000390 at human delta opioid receptors

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30 September 2017

Differential sorting of human delta-opioid receptors after internalization by peptide and alkaloid agonists.

1 reference

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30 September 2017

Endocytosis of the mu opioid receptor reduces tolerance and a cellular hallmark of opiate withdrawal

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2189997

30 September 2017

Mice deficient for delta- and mu-opioid receptors exhibit opposing alterations of emotional responses

1 reference

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30 September 2017

Internalization and recycling of delta-opioid receptor are dependent on a phosphorylation-dephosphorylation mechanism

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2189997

30 September 2017

Pharmacological delta1- and delta2-opioid receptor subtypes in the human neuroblastoma cell line SK-N-BE: no evidence for distinct molecular entities.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2189997

30 September 2017

Feedback inhibition of G protein-coupled receptor kinase 2 (GRK2) activity by extracellular signal-regulated kinases.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2189997

30 September 2017

Differential desensitization of human delta-opioid receptors by peptide and alkaloid agonists.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2189997

30 September 2017

Agonist-specific regulation of delta-opioid receptor trafficking by G protein-coupled receptor kinase and beta-arrestin

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2189997

30 September 2017

Opioid modulation of extracellular signal-regulated protein kinase activity is ras-dependent and involves Gbetagamma subunits

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2189997

30 September 2017

The delta-opioid receptor in SK-N-BE human neuroblastoma cell line undergoes heterologous desensitization

1 reference

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30 September 2017

The delta-opioid receptor regulates activity of ryanodine receptors in the human neuroblastoma cell line SK-N-BE.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2189997

30 September 2017

Loss of morphine-induced analgesia, reward effect and withdrawal symptoms in mice lacking the mu-opioid-receptor gene

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2189997

30 September 2017

delta- and mu-opioid receptor mobilization of intracellular calcium in SH-SY5Y human neuroblastoma cells

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2189997

30 September 2017

Morphine activates opioid receptors without causing their rapid internalization

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2189997

30 September 2017

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

1 reference

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30 September 2017

Behavioral despair in mice: a primary screening test for antidepressants

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30 September 2017

Phosphorylation and agonist-specific intracellular trafficking of an epitope-tagged mu-opioid receptor expressed in HEK 293 cells

1 reference

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30 September 2017

Convulsant activity of a non-peptidic delta-opioid receptor agonist is not required for its antidepressant-like effects in Sprague-Dawley rats

1 reference

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28 June 2018

Activity of the delta-opioid receptor is partially reduced, whereas activity of the kappa-receptor is maintained in mice lacking the mu-receptor.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2189997

28 June 2018

Opioid effects on mitogen-activated protein kinase signaling cascades

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2189997

28 June 2018

SK-N-BE: a human neuroblastoma cell line containing two subtypes of delta-opioid receptors.

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28 June 2018

Anxiolytic- and antidepressant-like activities of H-Dmt-Tic-NH-CH(CH2-COOH)-Bid (UFP-512), a novel selective delta opioid receptor agonist.

1 reference

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22 September 2018

Dmt-Tic-NH-CH2-Bid (UFP-502), a potent DOP receptor agonist: in vitro and in vivo studies.

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22 September 2018

Effects of the delta-opioid receptor agonist SNC80 on learning relative to its antidepressant-like effects in rats

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22 September 2018

Phosphorylation of activating transcription factor in murine splenocytes through delta opioid receptors

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22 September 2018

Potent delta-opioid receptor agonists containing the Dmt-Tic pharmacophore

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22 September 2018

Opioid receptor endocytosis and activation of MAP kinase pathway

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22 September 2018

Endogenous delta-opioid and ORL1 receptors couple to phosphorylation and activation of p38 MAPK in NG108-15 cells and this is regulated by protein kinase A and protein kinase C.

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22 September 2018

Synthesis and binding characteristics of [3H] H-Tyr-Ticpsi[CH2-NH] Cha-Phe-OH, a highly specific and stable delta-opioid antagonist

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22 September 2018

Desensitization of the delta-opioid receptor correlates with its phosphorylation in SK-N-BE cells: involvement of a G protein-coupled receptor kinase.

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22 September 2018

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10.1038/SJ.BJP.0707497

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9 January 2020

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9 January 2020

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