Rapid and efficient access to secondary arylmethylamines (Q36153388)

12 August 2017

Rapid and efficient access to secondary arylmethylamines (English)

1 reference

12 August 2017

Gary A Molander

1 reference

12 August 2017

Nicolas Fleury-Brégeot

1 reference

12 August 2017

Jessica Raushel

1 reference

12 August 2017

Deidre L Sandrock

1 reference

12 August 2017

Spencer D Dreher

1 reference

12 August 2017

language of work or name

English

0 references

publication date

5 July 2012

1 reference

Chemistry—A European Journal

12 August 2017

1 reference

12 August 2017

1 reference

12 August 2017

1 reference

12 August 2017

9564-9570

1 reference

Synthesis and cross-coupling reactions of imidomethyltrifluoroborates with aryl chlorides

12 August 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3415697

2 October 2017

Cross-coupling in flow

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3415697

Medicinal chemistry by the numbers: the physicochemistry, thermodynamics and kinetics of modern drug design.

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3415697

Synthesis and Cross-Coupling of Sulfonamidomethyltrifluoroborates

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3415697

Cross-Coupling of Mesylated Phenol Derivatives with Potassium Ammonio- and Amidomethyltrifluoroborates

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3415697

Synthesis of amidomethyltrifluoroborates and their use in cross-coupling reactions

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3415697

Aryl trifluoroborates in Suzuki-Miyaura coupling: the roles of endogenous aryl boronic acid and fluoride

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3415697

A convenient and general iron-catalyzed reduction of amides to amines

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3415697

The development of versatile methods for palladium-catalyzed coupling reactions of aryl electrophiles through the use of P(t-Bu)3 and PCy3 as ligands

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3415697

Scaffold diversity of natural products: inspiration for combinatorial library design

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3415697

Potassium organotrifluoroborates: new perspectives in organic synthesis.

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3415697

Organotrifluoroborates: protected boronic acids that expand the versatility of the Suzuki coupling reaction

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3415697

Synthesis of functionalized organotrifluoroborates via halomethyltrifluoroborates

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3415697

The evolving role of natural products in drug discovery

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3415697

Palladium-catalyzed Suzuki-Miyaura cross-coupling reactions of potassium aryl- and heteroaryltrifluoroborates

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3415697

Reductive Amination of Aldehydes and Ketones with Sodium Triacetoxyborohydride. Studies on Direct and Indirect Reductive Amination Procedures(1).

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3415697

Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3415697

Synthesis and Suzuki–Miyaura Cross-Coupling Reactions of Potassium Boc-Protected Aminomethyltrifluoroborate with Aryl and Hetaryl Halides

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3415697

Reinvestigation of Aminomethyltrifluoroborates and Their Application in Suzuki−Miyaura Cross-Coupling Reactions

2 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3415697

A new palladium precatalyst allows for the fast Suzuki-Miyaura coupling reactions of unstable polyfluorophenyl and 2-heteroaryl boronic acids

2 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3415697

Nucleophilicities of primary and secondary amines in water

2 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3415697

Aminomethylations via cross-coupling of potassium organotrifluoroborates with aryl bromides

2 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3415697

Structure-activity relationship of furosemide-derived compounds as antagonists of cerebellum-specific GABA(A) receptors

2 July 2018

1 reference

https://api.crossref.org/works/10.1002%2FCHEM.201200831

Reductive Aminations of Carbonyl Compounds with Borohydride and Borane Reducing Agents

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCHEM.201200831

1,2,3-Triazole-boranes: stable and efficient reagents for ketone and aldehyde reductive amination in organic solvents or in water

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCHEM.201200831

Ruthenium‐Catalyzed Nitro and Nitrile Compounds Coupling with Alcohols: Alternative Route for N‐Substituted Amine Synthesis

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCHEM.201200831

Controlled and Chemoselective Reduction of Secondary Amides

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCHEM.201200831

Scope of aminomethylations via Suzuki-Miyaura cross-coupling of organotrifluoroborates

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCHEM.201200831

Scope and mechanism of palladium-catalyzed amination of five-membered heterocyclic halides

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCHEM.201200831

Efficient ligandless palladium-catalyzed Suzuki reactions of potassium aryltrifluoroborates.

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCHEM.201200831

A novel approach to 3-methylindoles by a Heck/cyclization/isomerization process.

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCHEM.201200831

A Review on the Use of Sodium Triacetoxyborohydride in the Reductive Amination of Ketones and Aldehydes

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCHEM.201200831

A Versatile Catalyst for Reductive Amination by Transfer Hydrogenation

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCHEM.201200831

Cross-coupling reactions of potassium alkyltrifluoroborates with aryl and 1-alkenyl trifluoromethanesulfonates

21 January 2018

1 reference

12 December 2020

Cesium effect: high chemoselectivity in direct N-alkylation of amines

1 reference

12 December 2020

Efficient Nickel-Mediated Intramolecular Amination of Aryl Chlorides

1 reference

12 December 2020

Hydrosilane reduction of tertiary carboxamides by iron carbonyl catalysts

1 reference

12 December 2020

Hydrogen autotransfer in the N-alkylation of amines and related compounds using alcohols and amines as electrophiles

1 reference

12 December 2020

Suzuki-Miyaura Cross-Coupling Reactions in Flow: Multistep Synthesis Enabled by a Microfluidic Extraction

1 reference

12 December 2020

Mild NonepimerizingN-Alkylation of Amines by Alcohols without Transition Metals

1 reference

12 December 2020

Continuous-flow synthesis of 3,3-disubstituted oxindoles by a palladium-catalyzed α-arylation/alkylation sequence

1 reference

12 December 2020

Suzuki-Miyaura cross-coupling of heteroaryl halides and arylboronic acids in continuous flow

1 reference

12 December 2020

Continuous-flow synthesis of biaryls enabled by multistep solid-handling in a lithiation/borylation/Suzuki-Miyaura cross-coupling sequence

1 reference

12 December 2020

Organotrifluoroborate Hydrolysis: Boronic Acid Release Mechanism and an Acid–Base Paradox in Cross-Coupling

1 reference

12 December 2020

A Convenient and General Method for Pd-Catalyzed Suzuki Cross-Couplings of Aryl Chlorides and Arylboronic Acids

1 reference

12 December 2020

Identifiers

DOI

10.1002/CHEM.201200831

1 reference

12 August 2017

1 reference

12 August 2017

PubMed publication ID

22767518

1 reference