Pharmacological characterization of GSK1004723, a novel, long-acting antagonist at histamine H(1) and H(3) receptors (Q35593062)

9 August 2017

title

Pharmacological characterization of GSK1004723, a novel, long-acting antagonist at histamine H(1) and H(3) receptors (English)

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9 August 2017

R J Slack

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9 August 2017

L J Russell

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9 August 2017

D A Hall

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9 August 2017

M A Luttmann

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9 August 2017

A J Ford

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9 August 2017

K A Saunders

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9 August 2017

S T Hodgson

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9 August 2017

H E Connor

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9 August 2017

C Browning

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9 August 2017

K L Clark

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9 August 2017

language of work or name

English

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publication date

1 November 2011

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British Journal of Pharmacology

9 August 2017

published in

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9 August 2017

volume

164

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9 August 2017

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9 August 2017

page(s)

1627-1641

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Treatment of congestion in upper respiratory diseases

9 August 2017

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GSK189254, a novel H3 receptor antagonist that binds to histamine H3 receptors in Alzheimer's disease brain and improves cognitive performance in preclinical models

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Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

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Changes in pH differently affect the binding properties of histamine H1 receptor antagonists

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Activation of histamine H3 receptors in human nasal mucosa inhibits sympathetic vasoconstriction

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12 December 2020

Noninvasive Measurement of Airway Responsiveness in Allergic Mice Using Barometric Plethysmography

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Histamine and the nasal vasculature: the influence of H1 and H2-histamine receptor antagonism

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10.1111/J.1476-5381.2011.01285.X

Identifiers

DOI

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9 August 2017

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9 August 2017

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