Binding of serotonin and N1-benzenesulfonyltryptamine-related analogs at human 5-HT6 serotonin receptors: receptor modeling studies (Q34737074)

29 June 2018

title

Binding of serotonin and N1-benzenesulfonyltryptamine-related analogs at human 5-HT6 serotonin receptors: receptor modeling studies (English)

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29 June 2018

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Małgorzata Dukat

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29 June 2018

Philip D Mosier

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29 June 2018

Renata Kolanos

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29 June 2018

Bryan L Roth

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29 June 2018

Richard A Glennon

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29 June 2018

language of work or name

English

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publication date

18 January 2008

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29 June 2018

Journal of Medicinal Chemistry

published in

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29 June 2018

volume

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29 June 2018

issue

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29 June 2018

page(s)

603-611

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29 June 2018

Binding of sulfonyl-containing arylalkylamines at human 5-HT6 serotonin receptors

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7 July 2018

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7 July 2018

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7 July 2018

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7 July 2018

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7 July 2018

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7 July 2018

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7 July 2018

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7 July 2018

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7 July 2018

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5-Chloro-N-(4-methoxy-3-piperazin-1-yl- phenyl)-3-methyl-2-benzothiophenesulfon- amide (SB-271046): a potent, selective, and orally bioavailable 5-HT6 receptor antagonist

7 July 2018

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Identification of residues in transmembrane regions III and VI that contribute to the ligand binding site of the serotonin 5-HT6 receptor.

7 July 2018

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Characterization of Ro 04-6790 and Ro 63-0563: potent and selective antagonists at human and rat 5-HT6 receptors

7 July 2018

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7 July 2018

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Interaction of Tryptamine and Ergoline Compounds with Threonine 196 in the Ligand Binding Site of the 5-Hydroxytryptamine6Receptor

7 July 2018

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7 July 2018

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Cloning, characterization, and chromosomal localization of a human 5-HT6 serotonin receptor

7 July 2018

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Comparative protein modelling by satisfaction of spatial restraints

7 July 2018

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CLUSTAL W: improving the sensitivity of progressive multiple sequence alignment through sequence weighting, position-specific gap penalties and weight matrix choice

7 July 2018

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Binding of typical and atypical antipsychotic agents to 5-hydroxytryptamine-6 and 5-hydroxytryptamine-7 receptors

7 July 2018

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7 July 2018

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7 July 2018

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Contributions of Conserved Serine Residues to the Interactions of Ligands with Dopamine D2 Receptors

7 July 2018

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Further studies on the binding of N1-substituted tryptamines at h5-HT6 receptors

7 July 2018

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Interaction of N1-unsubstituted and N1-benzenesulfonyltryptamines at h5-HT6 receptors

26 October 2018

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A three-dimensional pharmacophore model for 5-hydroxytryptamine6 (5-HT6) receptor antagonists.

26 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5994921

Possible differences in modes of agonist and antagonist binding at human 5-HT6 receptors

26 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5994921

The retinal conformation and its environment in rhodopsin in light of a new 2.2 A crystal structure

26 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5994921

Protein-based virtual screening of chemical databases. II. Are homology models of G-Protein Coupled Receptors suitable targets?

26 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5994921

Indole inhibitors of human nonpancreatic secretory phospholipase A2. 1. Indole-3-acetamides

26 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5994921

Molecular recognition of receptor sites using a genetic algorithm with a description of desolvation

26 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5994921

Identification of two serine residues involved in agonist activation of the beta-adrenergic receptor

26 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/18201064

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Differential ergoline and ergopeptine binding to 5-hydroxytryptamine2A receptors: ergolines require an aromatic residue at position 340 for high affinity binding

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/18201064

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1021/JM070910S

1 reference

29 June 2018

PMC publication ID

5994921

1 reference

29 June 2018

PubMed publication ID

18201064

1 reference

29 June 2018