Iclaprim, a novel diaminopyrimidine with potent activity on trimethoprim sensitive and resistant bacteria (Q34277300)

1 August 2017

title

Iclaprim, a novel diaminopyrimidine with potent activity on trimethoprim sensitive and resistant bacteria (English)

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1 August 2017

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https://api.crossref.org/works/10.1016/J.BMCL.2003.07.023

3 April 2024

pharmaceutical science

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Crossref

https://api.crossref.org/works/10.1016/J.BMCL.2003.07.023

3 April 2024

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https://api.crossref.org/works/10.1016/J.BMCL.2003.07.023

3 April 2024

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https://api.crossref.org/works/10.1016/J.BMCL.2003.07.023

3 April 2024

Peter Schneider

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1 August 2017

Stephen Hawser

series ordinal

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1 August 2017

Khalid Islam

series ordinal

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1 August 2017

language of work or name

English

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publication date

1 December 2003

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full work available at URL

1 August 2017

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inferred from page(s)

https://api.elsevier.com/content/article/PII:S0960894X03008837?httpAccept=text/xml

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Crossref

https://api.crossref.org/works/10.1016/J.BMCL.2003.07.023

https://api.elsevier.com/content/article/PII:S0960894X03008837?httpAccept=text/plain

3 April 2024

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Crossref

https://api.crossref.org/works/10.1016/J.BMCL.2003.07.023

Bioorganic & Medicinal Chemistry Letters

3 April 2024

published in

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1 August 2017

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1 August 2017

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1 August 2017

page(s)

4217-4221

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A biochemical approach to chemotherapy

1 August 2017

cites work

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https://api.crossref.org/works/10.1016/J.BMCL.2003.07.023

Dihydrofolate reductases as targets for inhibitors

3 April 2024

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Dihydrofolate reductases as targets for inhibitors

3 April 2024

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Phenotypic expression in E. coli of a DNA sequence coding for mouse dihydrofolate reductase

3 April 2024

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A 1H NMR study of the interactions and conformations of rationally designed brodimoprim analogues in complexes with Lactobacillus casei dihydrofolate reductase

3 April 2024

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Solution structure of a brodimoprim analogue in its complex with Lactobacillus casei dihydrofolate reductase

3 April 2024

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https://api.crossref.org/works/10.1016/J.BMCL.2003.07.023

Receptor-based design of dihydrofolate reductase inhibitors: comparison of crystallographically determined enzyme binding with enzyme affinity in a series of carboxy-substituted trimethoprim analogues

3 April 2024

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Molecular modelling of trimethoprim complexes of human wild-type and mutant dihydrofolate reductases: identification of two subsets of binding residues in the antifolate binding site

3 April 2024

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Quantitative structure-selectivity relationships. Comparison of the inhibition of Escherichia coli and bovine liver dihydrofolate reductase by 5-(substituted-benzyl)-2,4-diaminopyrimidines.

3 April 2024

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On the optimization of hydrophobic and hydrophilic substituent interactions of 2,4-diamino-5-(substituted-benzyl)pyrimidines with dihydrofolate reductase

3 April 2024

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A single amino acid substitution in Staphylococcus aureus dihydrofolate reductase determines trimethoprim resistance

3 April 2024

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Trimethoprim resistance transposon Tn4003 from Staphylococcus aureus encodes genes for a dihydrofolate reductase and thymidylate synthetase flanked by three copies of IS257.

3 April 2024

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Identical genes for trimethoprim-resistant dihydrofolate reductase from Staphylococcus aureus in Australia and central Europe

3 April 2024

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Pharmacophore mapping of a series of 2,4-diamino-5-deazapteridine inhibitors of Mycobacterium avium complex dihydrofolate reductase

3 April 2024

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Design, synthesis, computational prediction, and biological evaluation of ester soft drugs as inhibitors of dihydrofolate reductase from Pneumocystis carinii

3 April 2024

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Structural studies on bioactive compounds. 34. Design, synthesis, and biological evaluation of triazenyl-substituted pyrimethamine inhibitors of Pneumocystis carinii dihydrofolate reductase

3 April 2024

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Effects of various test media on the activities of 21 antimicrobial agents against Haemophilus influenzae

3 April 2024

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3 April 2024

Identifiers

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release_e75vbcs4t5awbn5dwlqinrm65i

1 August 2017

Fatcat ID

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Fatcat

https://api.fatcat.wiki/v0/release/e75vbcs4t5awbn5dwlqinrm65i

mapped directly with Wikidata item

24 November 2022

based on heuristic

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