Kinetic analysis of estrogen receptor/ligand interactions (Q34064957)

30 July 2017

title

Kinetic analysis of estrogen receptor/ligand interactions (English)

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30 July 2017

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Rebecca L Rich

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30 July 2017

Lise R Hoth

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30 July 2017

Kieran F Geoghegan

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30 July 2017

Thomas A Brown

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30 July 2017

Peter K LeMotte

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30 July 2017

Samuel P Simons

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30 July 2017

Preston Hensley

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30 July 2017

David G Myszka

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30 July 2017

language of work or name

English

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publication date

19 June 2002

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Proceedings of the National Academy of Sciences of the United States of America

30 July 2017

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inferred from page(s)

published in

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30 July 2017

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30 July 2017

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30 July 2017

page(s)

8562-8567

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Direct comparison of binding equilibrium, thermodynamic, and rate constants determined by surface- and solution-based biophysical methods

30 July 2017

cites work

1 reference

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High resolution screening of plant natural product extracts for estrogen receptor alpha and beta binding activity using an online HPLC-MS biochemical detection system

5 July 2018

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Overexpression, purification, and crystal structure of native ER alpha LBD

5 July 2018

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Estrogen receptor-cofactor interactions as targets for novel drug discovery.

5 July 2018

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Structure-function evaluation of ER alpha and beta interplay with SRC family coactivators. ER selective ligands

5 July 2018

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Crystal structure of a mutant hERalpha ligand-binding domain reveals key structural features for the mechanism of partial agonism

5 July 2018

1 reference

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Differential effects of xenoestrogens on coactivator recruitment by estrogen receptor (ER) alpha and ERbeta.

5 July 2018

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5 July 2018

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Rational discovery of novel nuclear hormone receptor antagonists

5 July 2018

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EM-652 (SCH 57068), a third generation SERM acting as pure antiestrogen in the mammary gland and endometrium

5 July 2018

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Novel ligands that function as selective estrogens or antiestrogens for estrogen receptor-alpha or estrogen receptor-beta

5 July 2018

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Spontaneous α-N-6-Phosphogluconoylation of a “His Tag” inEscherichia coli:The Cause of Extra Mass of 258 or 178 Da in Fusion Proteins

5 July 2018

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The structural basis of estrogen receptor/coactivator recognition and the antagonism of this interaction by tamoxifen

5 July 2018

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Interaction of estrogenic chemicals and phytoestrogens with estrogen receptor beta

5 July 2018

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Rapid screening of environmental chemicals for estrogen receptor binding capacity

5 July 2018

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Discovery and preclinical pharmacology of a novel, potent, nonsteroidal estrogen receptor agonist/antagonist, CP-336156, a diaryltetrahydronaphthalene

5 July 2018

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Extending the range of rate constants available from BIACORE: interpreting mass transport-influenced binding data

5 July 2018

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Differential response of estrogen receptor alpha and estrogen receptor beta to partial estrogen agonists/antagonists

5 July 2018

1 reference

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Crystallographic comparison of the estrogen and progesterone receptor's ligand binding domains

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=124311

CLAMP: a biosensor kinetic data analysis program

5 July 2018

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Effects of CP-336,156, a new, nonsteroidal estrogen agonist/antagonist, on bone, serum cholesterol, uterus and body composition in rat models

5 July 2018

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Altered Ligand Binding Properties and Enhanced Stability of a Constitutively Active Estrogen Receptor: Evidence That an Open Pocket Conformation Is Required for Ligand Interaction

5 July 2018

1 reference

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Molecular basis of agonism and antagonism in the oestrogen receptor

5 July 2018

1 reference

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Comparison of the ligand binding specificity and transcript tissue distribution of estrogen receptors alpha and beta

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=124311

1,2-Diaryl-3,4-dihydronaphthalenes: photofluorogenic ligands for the estrogen receptor

5 July 2018

1 reference

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Estradiol- and estriol-binding in human benign prostatic hyperplasia

5 July 2018

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High-resolution and high-throughput protocols for measuring drug/human serum albumin interactions using BIACORE.

5 July 2018

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https://api.crossref.org/works/10.1073%2FPNAS.142288199

Transcriptional activities of estrogen receptor alpha and beta in yeast properties of raloxifene

21 January 2018

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https://api.crossref.org/works/10.1073%2FPNAS.142288199

Interactions of synthetic estrogens with human estrogen receptors

21 January 2018

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https://api.crossref.org/works/10.1073%2FPNAS.142288199

The estrogen receptor relative binding affinities of 188 natural and xenochemicals: structural diversity of ligands.

21 January 2018

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Differential SERM activation of the estrogen receptors (ERalpha and ERbeta) at AP-1 sites

21 January 2018

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Biosensor Analysis of the Interaction between Immobilized Human Serum Albumin and Drug Compounds for Prediction of Human Serum Albumin Binding Levels

21 January 2018

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https://api.crossref.org/works/10.1073%2FPNAS.142288199

Carboxylic acid analogues of tamoxifen: (Z)-2-[p-(1, 2-diphenyl-1-butenyl)phenoxy]-N,N-dimethylethylamine. Estrogen receptor affinity and estrogen antagonist effects in MCF-7 cells

21 January 2018

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12 December 2020

Structure-activity relationships of selective estrogen receptor modulators: modifications to the 2-arylbenzothiophene core of raloxifene

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12 December 2020

Improving biosensor analysis

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12 December 2020

Development of high throughput screening assays using fluorescence polarization: nuclear receptor-ligand-binding and kinase/phosphatase assays

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12 December 2020

Binding of xenobiotics to hepatic estrogen receptor and plasma sex steroid binding protein in the teleost fish, the common carp (Cyprinus carpio)

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12 December 2020

Receptor binding of NBD-labeled fluorescent estrogens and progestins in whole cells and cell-free preparations

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12 December 2020

Implementing surface plasmon resonance biosensors in drug discovery

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12 December 2020

Differential recruitment of the mammalian mediator subunit TRAP220 by estrogen receptors ERalpha and ERbeta

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12 December 2020

Binary quantitative structure-activity relationship (QSAR) analysis of estrogen receptor ligands

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12 December 2020

Identifiers

DOI

10.1073/PNAS.142288199

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30 July 2017

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30 July 2017

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