Pages that link to "Q39254269"

The following pages link to Dual-point competition association assay: a fast and high-throughput kinetic screening method for assessing ligand-receptor binding kinetics (Q39254269):

Displaying 24 items.

• A Four-Point Screening Method for Assessing Molecular Mechanism of Action (MMOA) Identifies Tideglusib as a Time-Dependent Inhibitor of Trypanosoma brucei GSK3β (Q28550557) (← links)
• New approaches for the reliable in vitro assessment of binding affinity based on high-resolution real-time data acquisition of radioligand-receptor binding kinetics (Q31172470) (← links)
• Mass spectrometry-based ligand binding assays on adenosine A1 and A2A receptors. (Q36289481) (← links)
• Drug-target residence time--a case for G protein-coupled receptors (Q38189272) (← links)
• Scintillation proximity assay (SPA) as a new approach to determine a ligand's kinetic profile. A case in point for the adenosine A1 receptor (Q38358474) (← links)
• Mechanistic models enable the rational use of in vitro drug-target binding kinetics for better drug effects in patients (Q38611990) (← links)
• Structure-Activity Relationships of the Sustained Effects of Adenosine A2A Receptor Agonists Driven by Slow Dissociation Kinetics. (Q38734217) (← links)
• Binding Kinetics in Drug Discovery (Q38918905) (← links)
• A novel CCR2 antagonist inhibits atherogenesis in apoE deficient mice by achieving high receptor occupancy (Q38936733) (← links)
• Structure-Affinity Relationships and Structure-Kinetics Relationships of Pyrido[2,1-f]purine-2,4-dione Derivatives as Human Adenosine A3 Receptor Antagonists (Q41722014) (← links)
• Molecular mechanism of allosteric modulation at GPCRs: insight from a binding kinetics study at the human A1 adenosine receptor (Q42221343) (← links)
• From receptor binding kinetics to signal transduction; a missing link in predicting in vivo drug-action (Q42620551) (← links)
• Structure-Affinity Relationships and Structure-Kinetic Relationships of 1,2-Diarylimidazol-4-carboxamide Derivatives as Human Cannabinoid 1 Receptor Antagonists (Q47103408) (← links)
• A binding kinetics study of human adenosine A3 receptor agonists. (Q47804733) (← links)
• Characterization of Kinetic Binding Properties of Unlabeled Ligands via a Preincubation Endpoint Binding Approach (Q50632046) (← links)
• Binding kinetics of ZM241385 derivatives at the human adenosine A2A receptor (Q51750607) (← links)
• Covalent Allosteric Probe for the Metabotropic Glutamate Receptor 2: Design, Synthesis, and Pharmacological Characterization. (Q52679428) (← links)
• A two-state model for the kinetics of competitive radioligand binding. (Q52683106) (← links)
• Evaluation of (4-Arylpiperidin-1-yl)cyclopentanecarboxamides As High-Affinity and Long-Residence-Time Antagonists for the CCR2 Receptor. (Q53481892) (← links)
• SNAPshots of the MCHR1: a Comparison Between the PET-Tracers [18F]FE@SNAP and [11C]SNAP-7941 (Q62862525) (← links)
• Probe dependency in the determination of ligand binding kinetics at a prototypical G protein-coupled receptor. (Q64944943) (← links)
• Route to Prolonged Residence Time at the Histamine H1 Receptor: Growing from Desloratadine to Rupatadine (Q91631033) (← links)
• Considerations for improved performance of competition association assays analysed with the Motulsky-Mahan's "kinetics of competitive binding" model (Q92837592) (← links)
• Binding pathway determines norepinephrine selectivity for the human β1AR over β2AR (Q100946468) (← links)