(Q39921218)

15 September 2017

A common intracellular allosteric binding site for antagonists of the CXCR2 receptor (English)

1 reference

15 September 2017

K Salchow

1 reference

15 September 2017

M E Bond

1 reference

15 September 2017

S C Evans

1 reference

15 September 2017

N J Press

1 reference

15 September 2017

S J Charlton

1 reference

15 September 2017

P A Hunt

1 reference

15 September 2017

M E Bradley

1 reference

15 September 2017

language of work or name

English

0 references

publication date

3 March 2010

1 reference

British Journal of Pharmacology

15 September 2017

1 reference

15 September 2017

159

1 reference

15 September 2017

1 reference

15 September 2017

1429-1439

1 reference

Chapter 12. The use of receptor homology modeling to facilitate the design of selective chemokine receptor antagonists

15 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2850400

Ligand binding and micro-switches in 7TM receptor structures

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2850400

CXCR2 antagonists for the treatment of pulmonary disease

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2850400

Identification of a putative intracellular allosteric antagonist binding-site in the CXC chemokine receptors 1 and 2.

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2850400

Allosteric inhibitors of chemoattractant receptors: opportunities and pitfalls

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2850400

An intracellular allosteric site for a specific class of antagonists of the CC chemokine G protein-coupled receptors CCR4 and CCR5.

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2850400

Pharmacological characterization of Sch527123, a potent allosteric CXCR1/CXCR2 antagonist

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2850400

The highly conserved DRY motif of class A G protein-coupled receptors: beyond the ground state.

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2850400

Allosterism at muscarinic receptors: ligands and mechanisms

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2850400

Noncompetitive allosteric inhibitors of the inflammatory chemokine receptors CXCR1 and CXCR2: prevention of reperfusion injury.

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2850400

Mutation of tyrosine in the conserved NPXXY sequence leads to constitutive phosphorylation and internalization, but not signaling, of the human B2 bradykinin receptor

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2850400

Differential roles of the NPXXY motif in formyl peptide receptor signaling

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2850400

A small region of the beta-adrenergic receptor is selectively involved in its rapid regulation

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2850400

SB265610 is an allosteric, inverse agonist at the human CXCR2 receptor

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2850400

Guide to Receptors and Channels (GRAC), 3rd edition

17 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2850400

Dual-function vector for protein expression in both mammalian cells and Xenopus laevis oocytes.

20 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2850400

Design of Noncompetitive Interleukin-8 Inhibitors Acting on CXCR1 and CXCR2

20 August 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20233217

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1111/J.1476-5381.2009.00623.X

1 reference

15 September 2017

1 reference

15 September 2017

PubMed publication ID

20233217

1 reference