(Q35685828)

English

2,3-Dihydro-1-benzofuran derivatives as a series of potent selective cannabinoid receptor 2 agonists: design, synthesis, and binding mode prediction through ligand-steered modeling.

scientific article published on October 2009

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3 February 2020

2,3-Dihydro-1-benzofuran derivatives as a series of potent selective cannabinoid receptor 2 agonists: design, synthesis, and binding mode prediction through ligand-steered modeling (English)

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3 February 2020

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cannabinoid receptor

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Claudio N. Cavasotto

7

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3 February 2020

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Philippe Diaz

1

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3 February 2020

Sharangdhar S Phatak

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3 February 2020

Jijun Xu

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3 February 2020

Frank R Fronczek

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3 February 2020

Fanny Astruc-Diaz

5

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3 February 2020

Charles M Thompson

6

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3 February 2020

Mohamed Naguib

8

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3 February 2020

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1 October 2009

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3 February 2020

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3 February 2020

4

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3 February 2020

10

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3 February 2020

1615-1629

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1 reference

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1 reference

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1 reference

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1 reference

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1 reference

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1 reference

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Design and synthesis of a novel series of N-alkyl isatin acylhydrazone derivatives that act as selective cannabinoid receptor 2 agonists for the treatment of neuropathic pain

1 reference

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1 reference

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1 reference

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1 reference

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1 reference

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1 reference

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1 reference

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1 reference

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12 July 2018

In vitro and in vivo characterization of A-796260: a selective cannabinoid CB2 receptor agonist exhibiting analgesic activity in rodent pain models

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3262993

12 July 2018

Targeting the cannabinoid CB2 receptor: modelling and structural determinants of CB2 selective ligands

1 reference

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12 July 2018

High-resolution crystal structure of an engineered human beta2-adrenergic G protein-coupled receptor

1 reference

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GPCR engineering yields high-resolution structural insights into beta2-adrenergic receptor function

1 reference

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12 July 2018

Crystal structure of the human beta2 adrenergic G-protein-coupled receptor

1 reference

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12 July 2018

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1 reference

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12 July 2018

N-Alkylidenearylcarboxamides as new potent and selective CB(2) cannabinoid receptor agonists with good oral bioavailability

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3262993

12 July 2018

New 1,2,3,4-tetrahydropyrrolo[3,4-b]indole derivatives as selective CB2 receptor agonists

1 reference

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12 July 2018

Comparative protein structure modeling by combining multiple templates and optimizing sequence-to-structure alignments.

1 reference

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12 July 2018

Sulfonamide derivatives as new potent and selective CB2 cannabinoid receptor agonists

1 reference

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Naphthalen-1-yl-(4-pentyloxynaphthalen-1-yl)methanone: a potent, orally bioavailable human CB1/CB2 dual agonist with antihyperalgesic properties and restricted central nervous system penetration

1 reference

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12 July 2018

Attenuation of allergic contact dermatitis through the endocannabinoid system

1 reference

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Discovery of 2-[(2,4-dichlorophenyl)amino]-N-[(tetrahydro- 2H-pyran-4-yl)methyl]-4-(trifluoromethyl)- 5-pyrimidinecarboxamide, a selective CB2 receptor agonist for the treatment of inflammatory pain.

1 reference

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Spinal cannabinoid receptor type 2 activation reduces hypersensitivity and spinal cord glial activation after paw incision

1 reference

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Characterization of chronic constriction of the saphenous nerve, a model of neuropathic pain in mice showing rapid molecular and electrophysiological changes

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Stimulation of cannabinoid receptor 2 (CB2) suppresses microglial activation

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Peripheral nerve injury induces cannabinoid receptor 2 protein expression in rat sensory neurons.

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12 July 2018

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1 reference

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12 July 2018

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1 reference

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12 July 2018

Structure of a cannabinoid receptor and functional expression of the cloned cDNA

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25 September 2018

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25 September 2018

CB2 cannabinoid receptor mediation of antinociception.

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25 September 2018

Virtual screening of novel CB2 ligands using a comparative model of the human cannabinoid CB2 receptor.

1 reference

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25 September 2018

Representing receptor flexibility in ligand docking through relevant normal modes.

1 reference

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25 September 2018

Behavioral, pharmacological and molecular characterization of the saphenous nerve partial ligation: a new model of neuropathic pain

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3262993

25 September 2018

Determinants of retinoid X receptor transcriptional antagonism

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3262993

25 September 2018

Toward the active conformations of rhodopsin and the beta2-adrenergic receptor

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3262993

25 September 2018

Protein flexibility in ligand docking and virtual screening to protein kinases.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3262993

25 September 2018

Induction of CB2 receptor expression in the rat spinal cord of neuropathic but not inflammatory chronic pain models

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3262993

25 September 2018

A critical role for a tyrosine residue in the cannabinoid receptors for ligand recognition

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3262993

25 September 2018

Treatments for chronic pain associated with spinal cord injuries: many are tried, few are helpful

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3262993

25 September 2018

A painful peripheral neuropathy in the rat produced by the chemotherapeutic drug, paclitaxel

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3262993

25 September 2018

CB2 cannabinoid receptor-mediated peripheral antinociception

1 reference

https://pubmed.ncbi.nlm.nih.gov/19637157

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Pharmacological proteus?

1 reference

https://pubmed.ncbi.nlm.nih.gov/19637157

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Analgesic Effects of Fatty Acid Amide Hydrolase Inhibition in a Rat Model of Neuropathic Pain

1 reference

https://pubmed.ncbi.nlm.nih.gov/19637157

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Phylogenomic and chemotaxonomic analysis of the endocannabinoid system

1 reference

https://pubmed.ncbi.nlm.nih.gov/19637157

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Protean behavior by agonists: agonist-directed trafficking of receptor signaling

1 reference

https://pubmed.ncbi.nlm.nih.gov/19637157

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The difference between the CB(1) and CB(2) cannabinoid receptors at position 5.46 is crucial for the selectivity of WIN55212-2 for CB(2)

1 reference

https://pubmed.ncbi.nlm.nih.gov/19637157

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Scalaradial, a Dialdehyde-Containing Marine Metabolite That Causes an Unexpected Noncovalent PLA2 Inactivation

1 reference

https://pubmed.ncbi.nlm.nih.gov/19637157

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Development and validation of a 96-well equilibrium dialysis apparatus for measuring plasma protein binding

1 reference

https://pubmed.ncbi.nlm.nih.gov/19637157

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Homology models of the cannabinoid CB1 and CB2 receptors. A docking analysis study

1 reference

https://pubmed.ncbi.nlm.nih.gov/19637157

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The third transmembrane helix of the cannabinoid receptor plays a role in the selectivity of aminoalkylindoles for CB2, peripheral cannabinoid receptor

1 reference

https://pubmed.ncbi.nlm.nih.gov/19637157

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Tricyclic pyrazoles. 4. Synthesis and biological evaluation of analogues of the robust and selective CB2 cannabinoid ligand 1-(2',4'-dichlorophenyl)-6-methyl-N-piperidin-1-yl-1,4-dihydroindeno[1,2-c]pyrazole-3-carboxamide

1 reference

https://pubmed.ncbi.nlm.nih.gov/19637157

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Switching modes for G protein-coupled receptor activation

1 reference

https://pubmed.ncbi.nlm.nih.gov/19637157

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

An efficient and selective method for the preparation of iodophenols

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200900226

7 January 2021

based on heuristic

inferred from DOI database lookup

Palladium-catalyzed cascade allylation/carbopalladation/cross coupling: a novel three-component reaction for the synthesis of 3,3-disubstituted-2,3-dihydrobenzofurans

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200900226

7 January 2021

based on heuristic

inferred from DOI database lookup

Efficient synthetic approach to heterocycles possessing the 3,3-disubstituted-2,3-dihydrobenzofuran skeleton via diverse palladium-catalyzed tandem reactions

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200900226

7 January 2021

based on heuristic

inferred from DOI database lookup

Conformational Sampling of Protein Flexibility in Generalized Coordinates: Application to Ligand Docking

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200900226

7 January 2021

based on heuristic

inferred from DOI database lookup

Identifiers

10.1002/CMDC.200900226

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:19637157%20AND%20SRC:MED&resulttype=core&format=json

3 February 2020

release_dagzvc237zbm3idu647abzcqma

1 reference

https://api.fatcat.wiki/v0/release/dagzvc237zbm3idu647abzcqma

24 November 2022

based on heuristic

mapped directly with Wikidata item

PMC publication ID

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:19637157%20AND%20SRC:MED&resulttype=core&format=json

3 February 2020

PubMed publication ID

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:19637157%20AND%20SRC:MED&resulttype=core&format=json

3 February 2020

ResearchGate publication ID

0 references

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