(Q33516043)

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Synthesis and pharmacological characterization of [(125)I]MRS5127, a high affinity, selective agonist radioligand for the A3 adenosine receptor

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Europe PubMed Central

PubMed publication ID

27 July 2017

Synthesis and pharmacological characterization of [(125)I]MRS5127, a high affinity, selective agonist radioligand for the A3 adenosine receptor (English)

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Europe PubMed Central

PubMed publication ID

27 July 2017

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Sonia de Castro

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Sonia de Castro

4

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Kenneth A. Jacobson

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Kenneth A Jacobson

6

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author name string

John A Auchampach

1

1 reference

Europe PubMed Central

PubMed publication ID

27 July 2017

Elizabeth T Gizewski

2

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Europe PubMed Central

PubMed publication ID

27 July 2017

Tina C Wan

3

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Europe PubMed Central

PubMed publication ID

27 July 2017

Garth G Brown

5

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Europe PubMed Central

PubMed publication ID

27 July 2017

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publication date

14 November 2009

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Europe PubMed Central

PubMed publication ID

27 July 2017

Biochemical Pharmacology

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Europe PubMed Central

PubMed publication ID

27 July 2017

79

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Europe PubMed Central

PubMed publication ID

27 July 2017

7

1 reference

Europe PubMed Central

PubMed publication ID

27 July 2017

967-973

1 reference

Europe PubMed Central

PubMed publication ID

27 July 2017

Functionalized congeners of A3 adenosine receptor-selective nucleosides containing a bicyclo[3.1.0]hexane ring system.

1 reference

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21 June 2018

Synthesis and characterization of [76Br]-labeled high-affinity A3 adenosine receptor ligands for positron emission tomography

1 reference

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21 June 2018

Selective A(3) adenosine receptor antagonists derived from nucleosides containing a bicyclo[3.1.0]hexane ring system

1 reference

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21 June 2018

The A3 adenosine receptor agonist CF102 induces apoptosis of hepatocellular carcinoma via de-regulation of the Wnt and NF-kappaB signal transduction pathways.

1 reference

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21 June 2018

The A3 adenosine receptor agonist CF502 inhibits the PI3K, PKB/Akt and NF-kappaB signaling pathway in synoviocytes from rheumatoid arthritis patients and in adjuvant-induced arthritis rats

1 reference

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21 June 2018

Synthesis and pharmacological characterization of [(125)I]MRS1898, a high-affinity, selective radioligand for the rat A(3) adenosine receptor.

1 reference

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21 June 2018

Design of (N)-methanocarba adenosine 5'-uronamides as species-independent A3 receptor-selective agonists.

1 reference

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21 June 2018

Clinical evidence for utilization of the A3 adenosine receptor as a target to treat rheumatoid arthritis: data from a phase II clinical trial

1 reference

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21 June 2018

The A3 adenosine receptor agonist CP-532,903 [N6-(2,5-dichlorobenzyl)-3'-aminoadenosine-5'-N-methylcarboxamide] protects against myocardial ischemia/reperfusion injury via the sarcolemmal ATP-sensitive potassium channel

1 reference

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21 June 2018

A3 adenosine receptor signaling contributes to airway mucin secretion after allergen challenge

1 reference

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21 June 2018

Adenosine receptors as therapeutic targets

1 reference

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21 June 2018

N6-ethyl-2-alkynyl NECAs, selective human A3 adenosine receptor agonists

1 reference

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21 June 2018

The cross-species A3 adenosine-receptor antagonist MRS 1292 inhibits adenosine-triggered human nonpigmented ciliary epithelial cell fluid release and reduces mouse intraocular pressure

1 reference

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21 June 2018

The A3 adenosine receptor is highly expressed in tumor versus normal cells: potential target for tumor growth inhibition

1 reference

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21 June 2018

Modulation of adenosine receptor affinity and intrinsic efficacy in adenine nucleosides substituted at the 2-position

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2815200

21 June 2018

Exploring distal regions of the A3 adenosine receptor binding site: sterically constrained N6-(2-phenylethyl)adenosine derivatives as potent ligands.

1 reference

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21 June 2018

N6-Substituted adenosine derivatives: selectivity, efficacy, and species differences at A3 adenosine receptors

1 reference

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21 June 2018

Medicinal chemistry of adenosine A3 receptor ligands

1 reference

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21 June 2018

[(3)H]8-Ethyl-4-methyl-2-phenyl-(8R)-4,5,7,8-tetrahydro-1H-imidazo[2,1-i]-purin-5-one ([(3)H]PSB-11), a novel high-affinity antagonist radioligand for human A(3) adenosine receptors

1 reference

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21 June 2018

A(1) or A(3) adenosine receptors induce late preconditioning against infarction in conscious rabbits by different mechanisms

1 reference

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21 June 2018

[(3)H]MRE 3008F20: a novel antagonist radioligand for the pharmacological and biochemical characterization of human A(3) adenosine receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2815200

21 June 2018

Canine Mast Cell Adenosine Receptors: Cloning and Expression of the A3Receptor and Evidence that Degranulation Is Mediated by the A2BReceptor

1 reference

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21 June 2018

Activation of A3 adenosine receptors on human eosinophils elevates intracellular calcium

1 reference

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21 June 2018

125I-4-aminobenzyl-5'-N-methylcarboxamidoadenosine, a high affinity radioligand for the rat A3 adenosine receptor

1 reference

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21 June 2018

Adenosine A3 receptor stimulation and cerebral ischemia

1 reference

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21 June 2018

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

1 reference

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21 June 2018

Preparation and first evaluation of [(18)F]FE@SUPPY: a new PET tracer for the adenosine A(3) receptor.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2815200

31 October 2018

Overexpression of A3 adenosine receptor in peripheral blood mononuclear cells in rheumatoid arthritis: involvement of nuclear factor-kappaB in mediating receptor level.

1 reference

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31 October 2018

[3H]HEMADO--a novel tritiated agonist selective for the human adenosine A3 receptor

1 reference

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31 October 2018

Activation of adenosine A3 receptors reduces ischemic brain injury in rodents.

1 reference

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31 October 2018

ADOA3R as a therapeutic target in experimental colitis: proof by validated high-density oligonucleotide microarray analysis

1 reference

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31 October 2018

Adenosine receptors in colon carcinoma tissues and colon tumoral cell lines: focus on the A(3) adenosine subtype

1 reference

https://pubmed.ncbi.nlm.nih.gov/19917269

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Preparation of N-succinimidyl 3-[*I]iodobenzoate: an agent for the indirect radioiodination of proteins

1 reference

https://pubmed.ncbi.nlm.nih.gov/19917269

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Are A3 adenosine receptors expressed in the brain?

1 reference

https://pubmed.ncbi.nlm.nih.gov/19917269

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1016/J.BCP.2009.11.009

1 reference

Europe PubMed Central

PubMed publication ID

27 July 2017

PMC publication ID

1 reference

Europe PubMed Central

PubMed publication ID

27 July 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

27 July 2017

ResearchGate publication ID

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