Azapropazone
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Nonsteroidal anti-inflammatory drug (NSAID)
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Trade names | Rheumox |
AHFS/Drugs.com | International Drug Names |
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Pharmacokinetic data | |
Elimination half-life | 20 hours |
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ECHA InfoCard | 100.033.543 |
Chemical and physical data | |
Formula | C16H20N4O2 |
Molar mass | 300.362 g·mol−1 |
3D model (JSmol) | |
Chirality | Racemic mixture |
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Azapropazone is a nonsteroidal anti-inflammatory drug (NSAID). It is manufactured by Goldshield under the tradename Rheumox.[1]
It was available in the UK as a prescription-only drug, with restrictions due to certain contra-indications and side-effects.[2] Azopropazone has now been discontinued in the British National Formulary.
Azapropazone has a half-life of approximately 20 hours in humans and is not extensively metabolized.[3]
References
- ^ "Rheumox Capsules". South Africa Electronic Package Inserts. Archived from the original on 2008-05-15. Retrieved 2008-08-18.
- ^ "Azapropazone". Patient UK. Archived from the original on 12 April 2009.
- ^ Jones CJ (1976). "The pharmacology and pharmacokinetics of azapropazone - a review". Current Medical Research and Opinion. 4 (1): 3–16. doi:10.1185/03007997609109277. PMID 770078.
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