Synthesis and pre-clinical evaluation of a potential radiotracer for PET imaging of the dopamine D3 receptor. (Q64907797)

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English	Synthesis and pre-clinical evaluation of a potential radiotracer for PET imaging of the dopamine D3 receptor.	scientific article

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6097203

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title

Synthesis and pre-clinical evaluation of a potential radiotracer for PET imaging of the dopamine D3 receptor (English)

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6097203

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Megan N Stewart

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1

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Peter J. H. Scott

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7

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Xia Shao

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2

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6097203

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Timothy J Desmond

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Taylor J Forrest

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4

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Janna Arteaga

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5

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Jenelle Stauff

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publication date

29 June 2018

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published in

MedChemComm

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9

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8

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1315-1322

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11C-labeling of n-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]arylcarboxamide derivatives and evaluation as potential radioligands for PET imaging of dopamine D3 receptors.

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18F-Labeled FAUC 346 and BP 897 derivatives as subtype-selective potential PET radioligands for the dopamine D3 receptor.

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Synthesis of new carbon-11-labeled carboxamide derivatives as potential PET dopamine D3 receptor radioligands

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Dopamine D3 receptor antagonists: the quest for a potentially selective PET ligand. Part one: lead identification.

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Dopamine D3 receptor antagonists: the quest for a potentially selective PET ligand. Part 3: Radiosynthesis and in vivo studies.

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High-affinity dopamine D2/D3 PET radioligands 18F-fallypride and 11C-FLB457: a comparison of kinetics in extrastriatal regions using a multiple-injection protocol

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[3H]4-(dimethylamino)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl) butyl)benzamide: a selective radioligand for dopamine D(3) receptors. II. Quantitative analysis of dopamine D(3) and D(2) receptor density ratio in the caudate-putamen

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Biodistribution studies of two 18F-labeled pyridinylphenyl amides as subtype selective radioligands for the dopamine D3 receptor

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Synthesis and evaluation of fluoro substituted pyridinylcarboxamides and their phenylazo analogues for potential dopamine D3 receptor PET imaging.

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Dopamine receptors - IUPHAR Review 13

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Dopamine D3 receptor binding of (18)F-fallypride: Evaluation using in vitro and in vivo PET imaging studies.

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Optimization and synthesis of an18F-labeled dopamine D3receptor ligand using [18F]fluorophenylazocarboxylictert-butylester

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Improving selectivity of dopamine D3 receptor ligands

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Synthesis of Diverse (11)C-Labeled PET Radiotracers via Direct Incorporation of [(11)C]CO2.

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The dopamine D3 receptor, a quarter century later.

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Absorbed radiation dosimetry of the D3-specific PET radioligand [18F]FluorTriopride estimated using rodent and nonhuman primate

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Small Molecule Receptor Ligands for PET Studies of the Central Nervous System-Focus on G Protein Coupled Receptors

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Identifiers

DOI

10.1039/C8MD00094H

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6097203

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PMC publication ID

6097203

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PMC publication ID

6097203

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PubMed publication ID

30151086

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PMC publication ID

6097203

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