Structure-Activity Relationship of Hetarylpropylguanidines Aiming at the Development of Selective Histamine Receptor Ligands (Q64061747)

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English	Structure-Activity Relationship of Hetarylpropylguanidines Aiming at the Development of Selective Histamine Receptor Ligands	article

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6401531

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29 April 2020

title

Structure-Activity Relationship of Hetarylpropylguanidines Aiming at the Development of Selective Histamine Receptor Ligands† (English)

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6401531

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29 April 2020

author

Steffen Pockes

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1

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6401531

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29 April 2020

David Wifling

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2

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6401531

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29 April 2020

Armin Buschauer

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3

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6401531

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29 April 2020

author name string

Sigurd Elz

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4

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6401531

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language of work or name

English

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publication date

5 March 2019

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6401531

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29 April 2020

published in

ChemistryOpen

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6401531

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volume

8

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6401531

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29 April 2020

issue

3

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6401531

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29 April 2020

page(s)

285-297

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6401531

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Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

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Selective ligands as tools to study histamine receptors

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Molecular cloning and characterization of a novel type of histamine receptor preferentially expressed in leukocytes

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Cloning and pharmacological characterization of a fourth histamine receptor (H(4)) expressed in bone marrow

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Cloning, expression, and pharmacological characterization of a novel human histamine receptor.

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Cloning and characterization of a novel human histamine receptor

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Histamine H3-receptor-mediated [35S]GTP gamma[S] binding: evidence for constitutive activity of the recombinant and native rat and human H3 receptors.

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Coordination of histamine H3 receptor antagonists with human adrenal cytochrome P450 enzymes

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Some chemical and physical properties associated with histamine antagonism

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N(G)-acylated imidazolylpropylguanidines as potent histamine H4 receptor agonists: selectivity by variation of the N(G)-substituent.

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New substructure filters for removal of pan assay interference compounds (PAINS) from screening libraries and for their exclusion in bioassays

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Promiscuous 2-aminothiazoles (PrATs): a frequent hitting scaffold.

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Histamine H3 receptor as a potential target for cognitive symptoms in neuropsychiatric diseases

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The dual-acting AChE inhibitor and H3 receptor antagonist UW-MD-72 reverses amnesia induced by scopolamine or dizocilpine in passive avoidance paradigm in rats

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The magnificent two: histamine and the H3 receptor as key modulators of striatal circuitry

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Histamine H3R receptor activation in the dorsal striatum triggers stereotypies in a mouse model of tic disorders

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The Ecstasy and Agony of Assay Interference Compounds

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Radiolabeled Dibenzodiazepinone-Type Antagonists Give Evidence of Dualsteric Binding at the M2 Muscarinic Acetylcholine Receptor.

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Highly Potent, Stable, and Selective Dimeric Hetarylpropylguanidine-Type Histamine H2 Receptor Agonists

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Identifiers

DOI

10.1002/OPEN.201900011

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Europe PubMed Central

PMC publication ID

6401531

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:30886786%20AND%20SRC:MED&resulttype=core&format=json

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29 April 2020

PMC publication ID

6401531

1 reference

stated in

Europe PubMed Central

PMC publication ID

6401531

reference URL

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:30886786%20AND%20SRC:MED&resulttype=core&format=json

retrieved

29 April 2020

PubMed publication ID

30886786

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stated in

Europe PubMed Central

PMC publication ID

6401531

reference URL

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:30886786%20AND%20SRC:MED&resulttype=core&format=json

retrieved

29 April 2020

 

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