Antagonist activities of mecamylamine and nicotine show reciprocal dependence on beta subunit sequence in the second transmembrane domain (Q35566473)

8 August 2017

title

Antagonist activities of mecamylamine and nicotine show reciprocal dependence on beta subunit sequence in the second transmembrane domain (English)

1 reference

8 August 2017

main subject

transmembrane protein

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author name string

J C Webster

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8 August 2017

M M Francis

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8 August 2017

J K Porter

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8 August 2017

G Robinson

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8 August 2017

C Stokes

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8 August 2017

B Horenstein

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8 August 2017

R L Papke

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8 August 2017

language of work or name

English

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publication date

1 July 1999

1 reference

British Journal of Pharmacology

8 August 2017

published in

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8 August 2017

volume

127

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8 August 2017

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8 August 2017

page(s)

1337-1348

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Sensitivity to voltage-independent inhibition determined by pore-lining region of the acetylcholine receptor

8 August 2017

cites work

1 reference

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Muscle-type nicotinic acetylcholine receptor delta subunit determines sensitivity to noncompetitive inhibitors, while gamma subunit regulates divalent permeability

12 July 2018

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12 July 2018

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12 July 2018

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12 July 2018

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12 July 2018

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12 July 2018

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12 July 2018

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12 July 2018

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12 July 2018

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12 July 2018

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12 July 2018

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12 July 2018

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12 July 2018

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12 July 2018

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12 July 2018

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12 July 2018

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12 July 2018

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26 September 2018

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Characterization of a series of anabaseine-derived compounds reveals that the 3-(4)-dimethylaminocinnamylidine derivative is a selective agonist at neuronal nicotinic alpha 7/125I-alpha-bungarotoxin receptor subtypes.

26 September 2018

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Agonist and antagonist effects of nicotine on chick neuronal nicotinic receptors are defined by alpha and beta subunits

26 September 2018

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A study of the desensitization produced by acetylcholine at the motor end-plate

26 September 2018

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12 December 2020

Agonist recognition site of the peripheral acetylcholine receptor ion channel complex differentiates the enantiomers of nicotine

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12 December 2020

Ganglionic blocking properties of 3-methylaminoisocamphane hydrochloride (mecamylamine): a secondary amine.

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12 December 2020

Neurotoxins distinguish between different neuronal nicotinic acetylcholine receptor subunit combinations

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12 December 2020

The acetylcholine receptor of the neuromuscular junction recognizes mecamylamine as a noncompetitive antagonist

1 reference

12 December 2020

Identifiers

DOI

10.1038/SJ.BJP.0702686

1 reference

8 August 2017

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8 August 2017

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