Potent selective nonpeptidic inhibitors of human lung tryptase. (Q35546388)

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10 December 2019

title

Potent selective nonpeptidic inhibitors of human lung tryptase (English)

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10 December 2019

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10 December 2019

L E Burgess

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10 December 2019

B J Newhouse

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10 December 2019

P Ibrahim

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10 December 2019

J Rizzi

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10 December 2019

M A Kashem

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10 December 2019

A Hartman

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10 December 2019

B J Brandhuber

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10 December 2019

C D Wright

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10 December 2019

D S Thomson

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10 December 2019

K Koch

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10 December 2019

language of work or name

English

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publication date

1 July 1999

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Proceedings of the National Academy of Sciences of the United States of America

10 December 2019

published in

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10 December 2019

volume

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10 December 2019

issue

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10 December 2019

page(s)

8348-8352

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On the attribution and additivity of binding energies

10 December 2019

cites work

1 reference

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1,2-Benzisothiazol-3-one 1,1-dioxide inhibitors of human mast cell tryptase.

12 July 2018

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A role for tryptase in the activation of human mast cells: modulation of histamine release by tryptase and inhibitors of tryptase

12 July 2018

1 reference

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Human beta-tryptase is a ring-like tetramer with active sites facing a central pore

12 July 2018

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Human mast cell tryptase: a stimulus of microvascular leakage and mast cell activation

12 July 2018

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Discovering high-affinity ligands for proteins: SAR by NMR

12 July 2018

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Purification, characterization and biological evaluation of recombinant leech-derived tryptase inhibitor (rLDTI) expressed at high level in the yeast Saccharomyces cerevisiae

12 July 2018

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The mast cells of the multiple sclerosis brain

12 July 2018

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Highly potent, selective, and low cost bis-tetrahydroaminacrine inhibitors of acetylcholinesterase. Steps toward novel drugs for treating Alzheimer's disease

12 July 2018

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Mast cell tryptase is a mitogen for epithelial cells. Stimulation of IL-8 production and intercellular adhesion molecule-1 expression

12 July 2018

1 reference

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Distribution, activation and tryptase/chymase phenotype of mast cells in the rheumatoid lesion

12 July 2018

1 reference

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Mast cells, cytokines, and metalloproteinases at the rheumatoid lesion: dual immunolocalisation studies

12 July 2018

1 reference

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Regulation of tryptase from human lung mast cells by heparin. Stabilization of the active tetramer

12 July 2018

1 reference

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The fibrinogenolytic activity of purified tryptase from human lung mast cells

12 July 2018

1 reference

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Synovial procollagenase activation by human mast cell tryptase dependence upon matrix metalloproteinase 3 activation

12 July 2018

1 reference

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Activation of pulmonary mast cells by bronchoalveolar allergen challenge. In vivo release of histamine and tryptase in atopic subjects with and without asthma

12 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=17520

Immunologic and physicochemical evidence for conformational changes occurring on conversion of human mast cell tryptase from active tetramer to inactive monomer. Production of monoclonal antibodies recognizing active tryptase.

12 July 2018

1 reference

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Degradation of Airway Neuropeptides by Human Lung Tryptase

12 July 2018

1 reference

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12 July 2018

New aspects of asthma

1 reference

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Pericellular substrates of human mast cell tryptase: 72,000 dalton gelatinase and fibronectin

12 July 2018

1 reference

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Induction of vascular permeability enhancement by human tryptase: dependence on activation of prekallikrein and direct release of bradykinin from kininogens.

12 July 2018

1 reference

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Bis(5-amidino-2-benzimidazolyl)methane and related amidines are potent, reversible inhibitors of mast cell tryptases.

26 September 2018

1 reference

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Rapid chromatographic technique for preparative separations with moderate resolution

26 September 2018

1 reference

Crossref

https://api.crossref.org/works/10.1073%2FPNAS.96.15.8348

The 1997 Asthma Management Guidelines and therapeutic issues relating to the treatment of asthma. National Heart, Lung, and Blood Institute

21 January 2018

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12 December 2020

[Effect of trypsin inhibitors on protein-bound trypsin]

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12 December 2020

Mast cell responses in rheumatoid synovium. Association of the MCTC subset with matrix turnover and clinical progression

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12 December 2020

Effect of human mast cell tryptase on human plasma proenzymes

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12 December 2020

Tryptase in nasal fluid is a useful marker of allergic rhinitis

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12 December 2020

Mast cell tryptase and chymase are potential regulators of neurogenic inflammation in psoriatic skin

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12 December 2020

Studies on the active center of trypsin. Further characterization of the hydrophobic binding site

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12 December 2020

Irreversible Enzyme Inhibitors. CVI.1 Proteolytic Enzymes. I. Bulk Tolerances in Trypsin-Inhibitor Complexes2

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12 December 2020

Preliminary study of the tryptase levels in the synovial fluid of patients with inflammatory arthritis

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12 December 2020

Granulocyte recruitment by human mast cell tryptase

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12 December 2020

Mast cell tryptase potentiates histamine-induced contraction in human sensitized bronchus

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12 December 2020

Identifiers

DOI

10.1073/PNAS.96.15.8348

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10411878%20AND%20SRC:MED&resulttype=core&format=json

10 December 2019

0 references

1 reference

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10 December 2019

PubMed publication ID

10411878

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10411878%20AND%20SRC:MED&resulttype=core&format=json