Use of the triazolotriazine [3H]ZM 241385 as a radioligand at recombinant human A2B adenosine receptors (Q28343854)

21 June 2017

title

Use of the triazolotriazine [3H]ZM 241385 as a radioligand at recombinant human A2B adenosine receptors (English)

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21 June 2017

X D Ji

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21 June 2017

K A Jacobson

series ordinal

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21 June 2017

language of work or name

English

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publication date

1 November 1999

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Drug design and discovery

21 June 2017

published in

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21 June 2017

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21 June 2017

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21 June 2017

page(s)

217-226

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Structure-activity relationships and molecular modeling of 3, 5-diacyl-2,4-dialkylpyridine derivatives as selective A3 adenosine receptor antagonists

21 June 2017

cites work

1 reference

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Characterization of the human brain putative A2B adenosine receptor expressed in Chinese hamster ovary (CHO.A2B4) cells

20 March 2017

1 reference

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125I-4-(2-[7-amino-2-[2-furyl][1,2,4]triazolo[2,3-a][1,3,5] triazin-5-yl-amino]ethyl)phenol, a high affinity antagonist radioligand selective for the A2a adenosine receptor

20 March 2017

1 reference

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Positive modulation of intracellular Ca2+ levels by adenosine A2b receptors, prostacyclin, and prostaglandin E1 via a cholera toxin-sensitive mechanism in human erythroleukemia cells

20 March 2017

1 reference

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The A2b adenosine receptor mediates cAMP responses to adenosine receptor agonists in human intestinal epithelia

20 March 2017

1 reference

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Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

20 March 2017

1 reference

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Canine Mast Cell Adenosine Receptors: Cloning and Expression of the A3Receptor and Evidence that Degranulation Is Mediated by the A2BReceptor

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3425640

The in vitro pharmacology of ZM 241385, a potent, non‐xanthine, A2a selective adenosine receptor antagonist

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3425640

Functionalized congeners of 1,3-dialkylxanthines: preparation of analogues with high affinity for adenosine receptors

29 September 2017

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Molecular cloning and expression of the cDNA for a novel A2-adenosine receptor subtype.

29 September 2017

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A2A adenosine receptors from rat striatum and rat pheochromocytoma PC12 cells: characterization with radioligand binding and by activation of adenylate cyclase

29 September 2017

1 reference

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Derivatives of the triazoloquinazoline adenosine antagonist (CGS 15943) having high potency at the human A2B and A3 receptor subtypes.

29 September 2017

1 reference

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2 June 2018

Adenosine A2B receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3425640

An endogenous A2B adenosine receptor coupled to cyclic AMP generation in human embryonic kidney (HEK 293) cells

2 June 2018

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Functional characterization of the A2b adenosine receptor in NIH 3T3 fibroblasts

2 June 2018

1 reference

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Adenosine receptor activation in human fibroblasts: nucleoside agonists and antagonists

2 June 2018

1 reference

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Adenosine antagonism by purines, pteridines and benzopteridines in human fibroblasts

2 June 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/10624567

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Subclasses of adenosine receptors in the central nervous system: Interaction with caffeine and related methylxanthines

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/10624567

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

PMC publication ID

3425640

0 references

1 reference