Structural insights into the mode of action of a pure antiestrogen (Q27630646)

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5 November 2019

title

Structural insights into the mode of action of a pure antiestrogen (English)

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5 November 2019

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5 November 2019

A M Brzozowski

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5 November 2019

J Walton

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5 November 2019

R E Hubbard

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5 November 2019

A G Thorsell

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5 November 2019

Y L Li

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5 November 2019

J A Gustafsson

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5 November 2019

M Carlquist

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5 November 2019

publication date

1 February 2001

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5 November 2019

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5 November 2019

volume

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5 November 2019

issue

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5 November 2019

page(s)

145-153

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The steroid and thyroid hormone receptor superfamily

5 November 2019

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Novel steroidal pure antiestrogens

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7 January 2021

Response to a specific antioestrogen (ICI 182780) in tamoxifen-resistant breast cancer

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Estrogen receptor (ER) modulators each induce distinct conformational changes in ER alpha and ER beta.

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7 January 2021

Inhibition of estrogen receptor-DNA binding by the "pure" antiestrogen ICI 164,384 appears to be mediated by impaired receptor dimerization

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7 January 2021

Antiestrogen ICI 164,384 reduces cellular estrogen receptor content by increasing its turnover

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7 January 2021

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7 January 2021

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7 January 2021

Molecular basis of agonism and antagonism in the oestrogen receptor

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7 January 2021

The structural basis of estrogen receptor/coactivator recognition and the antagonism of this interaction by tamoxifen

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7 January 2021

Structure of the ligand-binding domain of oestrogen receptor beta in the presence of a partial agonist and a full antagonist

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7 January 2021

Crystallographic comparison of the estrogen and progesterone receptor's ligand binding domains

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7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

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Identifiers

DOI

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5 November 2019

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