Structure-based design, synthesis, and biochemical and pharmacological characterization of novel salvinorin A analogues as active state probes of the kappa-opioid receptor (Q24646341)

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English	Structure-based design, synthesis, and biochemical and pharmacological characterization of novel salvinorin A analogues as active state probes of the kappa-opioid receptor	scientific article

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1 February 2020

Structure-based design, synthesis, and biochemical and pharmacological characterization of novel salvinorin A analogues as active state probes of the kappa-opioid receptor (English)

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1 February 2020

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Jordan Zjawiony

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1 February 2020

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Feng Yan

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Ruslan V Bikbulatov

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Viorel Mocanu

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Nedyalka Dicheva

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Carol E Parker

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William C Wetsel

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Philip D Mosier

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Richard B Westkaemper

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John A Allen

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Bryan L Roth

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1 July 2009

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6898-6908

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1 February 2020

Salvinorin A: a potent naturally occurring nonnitrogenous kappa opioid selective agonist

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7 April 2017

The conserved cysteine 7.38 residue is differentially accessible in the binding-site crevices of the mu, delta, and kappa opioid receptors

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7 April 2017

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27 September 2017

A graph-theory algorithm for rapid protein side-chain prediction

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7 April 2017

Ribosomal S6 kinase 2 directly phosphorylates the 5-hydroxytryptamine 2A (5-HT2A) serotonin receptor, thereby modulating 5-HT2A signaling

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27 September 2017

Conformational changes involved in G-protein-coupled-receptor activation

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27 September 2017

Salvinorin A analogs as probes in opioid pharmacology

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27 September 2017

Galpha-subunits differentially alter the conformation and agonist affinity of kappa-opioid receptors

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27 September 2017

Wide turn diversity in protein transmembrane helices implications for G-protein-coupled receptor and other polytopic membrane protein structure and function.

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A clickable inhibitor reveals context-dependent autoactivation of p90 RSK

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27 September 2017

Differential helical orientations among related G protein-coupled receptors provide a novel mechanism for selectivity. Studies with salvinorin A and the kappa-opioid receptor

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27 September 2017

An opioid agonist that does not induce mu-opioid receptor--arrestin interactions or receptor internalization

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27 September 2017

Salvinorin A: from natural product to human therapeutics

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27 September 2017

Antinociceptive and hypothermic effects of Salvinorin A are abolished in a novel strain of kappa-opioid receptor-1 knockout mice

1 reference

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27 September 2017

The seventh transmembrane domains of the delta and kappa opioid receptors have different accessibility patterns and interhelical interactions

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27 September 2017

Determination of salvinorins and divinatorins in Salvia divinorum leaves by liquid chromatography/multistage mass spectrometry

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27 September 2017

Neoclerodane diterpenes as a novel scaffold for mu opioid receptor ligands.

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27 September 2017

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27 September 2017

Salvinorin A: the "magic mint" hallucinogen finds a molecular target in the kappa opioid receptor

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27 September 2017

Identification by MALDI-TOF mass spectrometry of 17 alpha-bromoacetamidopropylestradiol covalent attachment sites on estrogen receptor alpha.

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Hinges, swivels and switches: the role of prolines in signalling via transmembrane alpha-helices

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27 September 2017

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27 September 2017

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27 September 2017

Proximity-accelerated chemical coupling reaction in the benzodiazepine-binding site of gamma-aminobutyric acid type A receptors: superposition of different allosteric modulators.

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30 May 2018

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30 May 2018

[3H]beta-funaltrexamine binds covalently to brain opioid receptors

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30 May 2018

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30 May 2018

Synthetic studies of neoclerodane diterpenes from Salvia divinorum: preparation and opioid receptor activity of salvinicin analogues

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28 November 2018

Identification of the molecular mechanisms by which the diterpenoid salvinorin A binds to kappa-opioid receptors

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10.1021/BI900605N

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