Pharmacophore-based discovery of ligands for drug transporters (Q35594214)

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scientific article published on 26 September 2006

Language	Label	Description	Also known as
English	Pharmacophore-based discovery of ligands for drug transporters	scientific article published on 26 September 2006

Statements

scholarly article

1 reference

Europe PubMed Central

PubMed publication ID

9 August 2017

1 reference

Europe PubMed Central

Pharmacophore-based discovery of ligands for drug transporters (English)

1 reference

Europe PubMed Central

PubMed publication ID

9 August 2017

2

1 reference

Europe PubMed Central

PubMed publication ID

9 August 2017

object named as

Peter W Swaan

4

0 references

author name string

Cheng Chang

1

1 reference

Europe PubMed Central

PubMed publication ID

9 August 2017

Praveen Bahadduri

3

1 reference

Europe PubMed Central

PubMed publication ID

9 August 2017

language of work or name

0 references

publication date

26 September 2006

1 reference

Europe PubMed Central

PubMed publication ID

9 August 2017

Advanced Drug Delivery Reviews

1 reference

Europe PubMed Central

PubMed publication ID

9 August 2017

58

1 reference

Europe PubMed Central

PubMed publication ID

9 August 2017

12-13

1 reference

Europe PubMed Central

PubMed publication ID

9 August 2017

1431-1450

1 reference

Europe PubMed Central

PubMed publication ID

9 August 2017

Comparison of drug transporter levels in normal colon, colon cancer, and Caco-2 cells: impact on drug disposition and discovery.

1 reference

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Synthesis and Ligand Binding Studies of 4‘-Iodobenzoyl Esters of Tropanes and Piperidines at the Dopamine Transporter

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1773055

26 September 2018

A genetic algorithm for flexible molecular overlay and pharmacophore elucidation.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1773055

26 September 2018

A fast new approach to pharmacophore mapping and its application to dopaminergic and benzodiazepine agonists.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1773055

26 September 2018

Genetically evolved receptor models: a computational approach to construction of receptor models.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1773055

26 September 2018

Compass: predicting biological activities from molecular surface properties. Performance comparisons on a steroid benchmark

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1773055

26 September 2018

Validation of a Caco-2 cell monolayer culture for drug transport studies

1 reference

https://pubmed.ncbi.nlm.nih.gov/17097188

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

CHO/hPEPT1 cells overexpressing the human peptide transporter (hPEPT1) as an alternative in vitro model for peptidomimetic drugs

1 reference

https://pubmed.ncbi.nlm.nih.gov/17097188

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Role of breast cancer resistance protein in the bioavailability and fetal penetration of topotecan

1 reference

https://pubmed.ncbi.nlm.nih.gov/17097188

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Cellular uptake mechanism of amino acid ester prodrugs in Caco-2/hPEPT1 cells overexpressing a human peptide transporter

1 reference

https://pubmed.ncbi.nlm.nih.gov/17097188

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Transport of glutathione, glucuronate, and sulfate conjugates by the MRP gene-encoded conjugate export pump

1 reference

https://pubmed.ncbi.nlm.nih.gov/17097188

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Determination of in vitro permeability of drug candidates through a caco-2 cell monolayer by liquid chromatography/tandem mass spectrometry

1 reference

https://pubmed.ncbi.nlm.nih.gov/17097188

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Comparison of intestinal permeabilities determined in multiple in vitro and in situ models: relationship to absorption in humans

1 reference

https://pubmed.ncbi.nlm.nih.gov/17097188

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

A novel approach to predicting P450 mediated drug metabolism. CYP2D6 catalyzed N-dealkylation reactions and qualitative metabolite predictions using a combined protein and pharmacophore model for CYP2D6

1 reference

https://pubmed.ncbi.nlm.nih.gov/17097188

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Characterization of Caco-2 cell monolayer drug transport properties by cassette dosing using UV/fluorescence HPLC

1 reference

https://pubmed.ncbi.nlm.nih.gov/17097188

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The significance of peptides in clinical nutrition

1 reference

https://pubmed.ncbi.nlm.nih.gov/17097188

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Absorption of ACE inhibitors from small intestine and colon

1 reference

https://pubmed.ncbi.nlm.nih.gov/17097188

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Evidence for overlapping substrate specificity between large neutral amino acid (LNAA) and dipeptide (hPEPT1) transporters for PD 158473, an NMDA antagonist

1 reference

https://pubmed.ncbi.nlm.nih.gov/17097188

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

P-glycoprotein inhibitor erythromycin increases oral bioavailability of talinolol in humans

1 reference

https://pubmed.ncbi.nlm.nih.gov/17097188

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The product of the ABC half-transporter gene ABCG2 (BCRP/MXR/ABCP) is expressed in the plasma membrane

1 reference

https://pubmed.ncbi.nlm.nih.gov/17097188

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Proton-cotransport of pravastatin across intestinal brush-border membrane

1 reference

https://pubmed.ncbi.nlm.nih.gov/17097188

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1016/J.ADDR.2006.09.006

1 reference

Europe PubMed Central

PubMed publication ID

9 August 2017

release_dvhdgppf3nbdbifobkrtofasmm

1 reference

https://api.fatcat.wiki/v0/release/dvhdgppf3nbdbifobkrtofasmm

24 November 2022

based on heuristic

mapped directly with Wikidata item

PMC publication ID

1 reference

Europe PubMed Central

PubMed publication ID

9 August 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

9 August 2017

ResearchGate publication ID

0 references

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