Structure-activity relationships for inhibition of cysteine protease activity and development of Plasmodium falciparum by peptidyl vinyl sulfones (Q34722632)

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English	Structure-activity relationships for inhibition of cysteine protease activity and development of Plasmodium falciparum by peptidyl vinyl sulfones	scientific article

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scholarly article

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Europe PubMed Central

PubMed publication ID

4 August 2017

Structure-activity relationships for inhibition of cysteine protease activity and development of Plasmodium falciparum by peptidyl vinyl sulfones (English)

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Europe PubMed Central

PubMed publication ID

4 August 2017

Plasmodium falciparum

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Philip J Rosenthal

8

object named as

Philip J Rosenthal

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Europe PubMed Central

PubMed publication ID

4 August 2017

author name string

Bhaskar R Shenai

1

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Europe PubMed Central

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4 August 2017

Belinda J Lee

2

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Europe PubMed Central

PubMed publication ID

4 August 2017

Alejandro Alvarez-Hernandez

3

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Europe PubMed Central

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4 August 2017

Pek Y Chong

4

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Europe PubMed Central

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4 August 2017

Cory D Emal

5

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Europe PubMed Central

PubMed publication ID

4 August 2017

R Jeffrey Neitz

6

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4 August 2017

William R Roush

7

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4 August 2017

language of work or name

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publication date

1 January 2003

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4 August 2017

Antimicrobial Agents and Chemotherapy

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Europe PubMed Central

PubMed publication ID

4 August 2017

47

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Europe PubMed Central

PubMed publication ID

4 August 2017

1

1 reference

Europe PubMed Central

PubMed publication ID

4 August 2017

154-160

1 reference

Europe PubMed Central

PubMed publication ID

4 August 2017

Cysteine proteases of parasitic organisms

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=149004

7 July 2018

Hydrolysis of erythrocyte proteins by proteases of malaria parasites

1 reference

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7 July 2018

Medical need, scientific opportunity and the drive for antimalarial drugs

1 reference

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The economic and social burden of malaria

1 reference

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7 July 2018

Four plasmepsins are active in the Plasmodium falciparum food vacuole, including a protease with an active-site histidine

1 reference

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Expression and characterization of the Plasmodium falciparum haemoglobinase falcipain-3

1 reference

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Active site mapping, biochemical properties and subcellular localization of rhodesain, the major cysteine protease of Trypanosoma brucei rhodesiense

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Potent second generation vinyl sulfonamide inhibitors of the trypanosomal cysteine protease cruzain

1 reference

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Rapid and general profiling of protease specificity by using combinatorial fluorogenic substrate libraries

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Synthesis and Biological Activity of a Series of Potent Fluoromethyl Ketone Inhibitors of Recombinant Human Calpain I

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7 July 2018

Hemoglobin metabolism in the malaria parasite Plasmodium falciparum

1 reference

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7 July 2018

Antimalarial effects of vinyl sulfone cysteine proteinase inhibitors

1 reference

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7 July 2018

Investigation of the substrate specificity of cruzipain, the major cysteine proteinase of Trypanosoma cruzi, through the use of cystatin-derived substrates and inhibitors

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7 July 2018

Inhibition of a Plasmodium vinckei cysteine proteinase cures murine malaria

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7 July 2018

The proteases and pathogenicity of parasitic protozoa

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Vinylogous amino acid esters: a new class of inactivators for thiol proteases

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7 July 2018

A malarial cysteine proteinase is necessary for hemoglobin degradation by Plasmodium falciparum

1 reference

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7 July 2018

Isolation and characterization of a cysteine proteinase gene of Plasmodium falciparum

1 reference

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Synchronization of Plasmodium falciparum Erythrocytic Stages in Culture

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Reducing requirements for hemoglobin hydrolysis by Plasmodium falciparum cysteine proteases

1 reference

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26 October 2018

Antimalarial effects in mice of orally administered peptidyl cysteine protease inhibitors

1 reference

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1 reference

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1 reference

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1 reference

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Orally active trifluoromethyl ketone inhibitors of human leukocyte elastase

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Identifiers

10.1128/AAC.47.1.154-160.2003

1 reference

Europe PubMed Central

PubMed publication ID

4 August 2017

PMC publication ID

1 reference

Europe PubMed Central

PubMed publication ID

4 August 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

4 August 2017

ResearchGate publication ID

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