CCK-B antagonists in the control of anxiety and gastric acid secretion. (Q33938906)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10845247%20AND%20SRC:MED&resulttype=core&format=json

7 November 2019

review article

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title

CCK-B antagonists in the control of anxiety and gastric acid secretion (English)

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7 November 2019

M S Chambers

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7 November 2019

S R Fletcher

series ordinal

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7 November 2019

publication date

1 January 2000

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Progress in medicinal chemistry

7 November 2019

published in

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7 November 2019

volume

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7 November 2019

page(s)

45-81

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Structure of porcine cholecystokinin-pancreozymin. 1. Cleavage with thrombin and with trypsin

7 November 2019

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The panicogenic effects of cholecystokinin-tetrapeptide are antagonized by L-365,260, a central cholecystokinin receptor antagonist, in patients with panic disorder

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The CCKB receptor antagonist, L-365,260, elicits antidepressant-type effects in the forced-swim test in mice

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A selective CCKB receptor antagonist potentiates, mu-, but not delta-opioid receptor-mediated antinociception in the formalin test

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Failure of CCK receptor ligands to modify anxiety-related behavioural suppression in an operant conflict paradigm in rats

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Gastrin is a major mediator of the gastric phase of acid secretion in dogs: proof by monoclonal antibody neutralization

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Effect of gastrin receptor antagonists on gastric acid secretion and gastrin and somatostatin release in the rat stomach

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Cholecystokinin-tetrapeptide induces panic attacks in patients with panic disorder

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Cholecystokinin and anxiety in normal volunteers: an investigation of the anxiogenic properties of pentagastrin and reversal by the cholecystokinin receptor subtype B antagonist L-365,260

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7 January 2021

Effect of CI-988 on cholecystokinin tetrapeptide-induced panic symptoms in healthy volunteers

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7 January 2021

A placebo-controlled trial of L-365,260, a CCKB antagonist, in panic disorder

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7 January 2021

The cholecystokinin-B receptor antagonist CI-988 failed to affect CCK-4 induced symptoms in panic disorder patients

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7 January 2021

Second Generation “Peptoid” CCK-B Receptor Antagonists: Identification and Development ofN-(Adamantyloxycarbonyl)-α-methyl-(R)-tryptophan Derivative (CI-1015) with an Improved Pharmacokinetic Profile

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7 January 2021

Characterization of antigastrin activity in vivo of CR 2194, a new R-4-benzamido-5-oxo-pentanoic acid derivative

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7 January 2021

The gastrin-receptor antagonist L-365,260 inhibits stimulated acid secretion in humans

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7 January 2021

Benzodiazepine gastrin and brain cholecystokinin receptor ligands: L-365,260.

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7 January 2021

Second-generation benzodiazepine CCK-B antagonists. Development of subnanomolar analogs with selectivity and water solubility

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7 January 2021

Measurement of central nervous system activity of systemically administered CCKB receptor antagonists by ex vivo binding

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7 January 2021

Controlled modification of acidity in cholecystokinin B receptor antagonists: N-(1,4-benzodiazepin-3-yl)-N'-[3-(tetrazol-5-ylamino) phenyl]ureas

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High-affinity and potent, water-soluble 5-amino-1,4-benzodiazepine CCKB/gastrin receptor antagonists containing a cationic solubilizing group

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7 January 2021

The cholecystokinin-B receptor antagonist L-740,093 produces an insurmountable antagonism of CCK-4 stimulated functional response in cells expressing the human CCK-B receptor

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5-(Piperidin-2-yl)- and 5-(Homopiperidin-2-yl)-1,4-benzodiazepines: High-Affinity, Basic Ligands for the Cholecystokinin-B Receptor

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Synthesis and Evaluation of 1,5-Benzodiazepines with Bridged Cycloalkyl Substituents at the N-1 Position as Potent and Selective CCK-B Ligands

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7 January 2021

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7 January 2021

Rationally designed "dipeptoid" analogues of CCK. alpha-Methyltryptophan derivatives as highly selective and orally active gastrin and CCK-B antagonists with potent anxiolytic properties

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7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

The use of receptor desensitization to analyse CCKA and CCKB/gastrin receptors coupled to contraction in guinea-pig stomach muscle

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7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

A single amino acid of the cholecystokinin-B/gastrin receptor determines specificity for non-peptide antagonists

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7 January 2021

Antipsychotic potential of CCK-based treatments: an assessment using the prepulse inhibition model of psychosis

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7 January 2021

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7 January 2021

CCK in anxiety and cognitive processes

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7 January 2021

The anxieties of drug discovery and development. CCK-B receptor antagonists

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7 January 2021

10.1016/S0079-6468(08)70057-2

Identifiers

DOI

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10845247%20AND%20SRC:MED&resulttype=core&format=json

7 November 2019

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